SCHEMBL3696360

SCHEMBL3696360

O=C(O)c1nc2c(C=Cc3ccccc3)cc(-c3ccccc3)cn2c1Cl

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
BCL2L1 Q07817 1/20 0.39
BAD Q92934 1/20 0.39
ATP4A P20648 2/20 0.36
ATP4B P51164 2/20 0.36
MDM2 Q00987 3/20 0.36
PTPN1 P18031 1/20 0.35
PTPN6 P29350 1/20 0.35
HDAC1 Q13547 1/20 0.34
PTGES O14684 1/20 0.34
CTRC Q99895 1/20 0.33
LDHA P00338 1/20 0.33
KDM4E B2RXH2 1/20 0.33
LMNA P02545 1/20 0.33
HTT P42858 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
HDAC2 Q92769 1/20 0.33
DHODH Q02127 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3696358 1.00 BCL2L1 (0.39) BCL2L1BADATP4AATP4BMDM2
SCHEMBL3695641 0.81 AKR1C2 (0.41) MDM2CTRC
SCHEMBL3688691 0.81 NPC1 (0.43) HDAC1L3MBTL1
SCHEMBL7499668 0.80 RAB9A (0.46) LMNAHTT
SCHEMBL3684406 0.79 AKR1C4 (0.39) MDM2PTPN1CTRCLDHADHODH
SCHEMBL3689623 0.78 LDHA (0.43) MDM2CTRCLDHAKDM4ELMNA
SCHEMBL3687772 0.76 KMT2A (0.36) PTPN1KDM4ELMNAHTT
SCHEMBL3687771 0.76 KMT2A (0.36) PTPN1KDM4ELMNAHTT
SCHEMBL3699155 0.73 SERPINE1 (0.36) MDM2PTPN1LMNA
SCHEMBL3687376 0.71 GRM2 (0.44)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120121540-A1 Certain Nitrogen Containing Bicyclic Chemical Entities For Treating Viral Infections GLAXOSMITHKLINE LLC 2012-05-17 US disclosed
EP-2187883-A2 NITROGEN CONTAINING BICYCLIC CHEMICAL ENTITIES FOR TREATING VIRAL INFECTIONS GENELABS TECHNOLOGIES, INC. (US) 2010-05-26 EP disclosed
US-20090176778-A1 Certain nitrogen containing bicyclic chemical entities for treating viral infections GLAXOSMITHKLINE LLC 2009-07-09 US disclosed
WO-2009023179-A2 NITROGEN CONTAINING BICYCLIC CHEMICAL ENTITIES FOR TREATING VIRAL INFECTIONS GENELABS TECHNOLOGIES, INC. (US) 2009-02-19 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120121540-A1 Certain Nitrogen Containing Bicyclic Chemical Entities For Treating Viral Infections OAT, HAVCR2, CPS1 BCL2L1 2398/4885BAD 547/4885ATP4A 2486/4885
US-20090176778-A1 Certain nitrogen containing bicyclic chemical entities for treating viral infections OAT, HAVCR2, CPS1 BCL2L1 2398/4885BAD 547/4885ATP4A 2486/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.