SCHEMBL3697752

SCHEMBL3697752

CC(C)(C)CN(Cc1cc(Sc2cccnc2)n(-c2cccc(F)c2Cl)n1)C(=O)O

nearest known ligand 0.32

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
GPBAR1 Q8TDU6 1/20 0.31
DAGLB Q8NCG7 1/20 0.31
DAGLA Q9Y4D2 1/20 0.31
NOS3 P29474 1/20 0.31
NOS1 P29475 1/20 0.31
NOS2 P35228 1/20 0.31
TP53 P04637 1/20 0.30
CACNA1G O43497 1/20 0.30
CACNA1H O95180 1/20 0.30
CACNA1I Q9P0X4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3702437 0.90 MDM2 (0.33) GPBAR1DAGLBDAGLA
SCHEMBL3700538 0.89
SCHEMBL3701902 0.88 SLC16A3 (0.38)
SCHEMBL4131517 0.87 GPBAR1 (0.33) ALDH1A1NPSR1GPBAR1NOS3NOS1
SCHEMBL3690717 0.87 ALDH1A1 (0.33) ALDH1A1NPSR1DAGLBDAGLA
SCHEMBL3697749 0.83 HTR2C (0.45) NPSR1GPBAR1
SCHEMBL3706681 0.82
SCHEMBL3703232 0.82 SLC16A3 (0.31)
SCHEMBL3692815 0.82 SCN9A (0.33) TP53
SCHEMBL3709568 0.82 SLC16A3 (0.33) ALDH1A1NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2190822-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2010-06-02 EP disclosed
WO-2009041705-A9 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL (JP) 2009-08-13 WO disclosed
WO-2009041705-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-04-02 WO disclosed