SCHEMBL3702437

SCHEMBL3702437

CC(C)(C)CN(Cc1cc(Sc2cccnc2)n(-c2cccc(Cl)c2F)n1)C(=O)O

nearest known ligand 0.33

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MDM2 Q00987 2/20 0.33
RIPK1 Q13546 1/20 0.33
NOTUM Q6P988 1/20 0.32
SLC16A3 O15427 2/20 0.31
SLC16A1 P53985 2/20 0.31
GPBAR1 Q8TDU6 1/20 0.31
DAGLB Q8NCG7 1/20 0.31
DAGLA Q9Y4D2 1/20 0.31
CFD P00746 1/20 0.30
USP2 O75604 1/20 0.30
TSHR P16473 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3701902 0.92 SLC16A3 (0.38) SLC16A3SLC16A1
SCHEMBL3706681 0.91
SCHEMBL3697752 0.90 ALDH1A1 (0.32) GPBAR1DAGLBDAGLA
SCHEMBL3690717 0.89 ALDH1A1 (0.33) DAGLBDAGLA
SCHEMBL3814318 0.89 MDM2 (0.33) MDM2RIPK1NOTUMSLC16A3SLC16A1
SCHEMBL4120305 0.87 MDM2 (0.36) MDM2RIPK1NOTUMSLC16A3SLC16A1
SCHEMBL3702432 0.83 HTR2C (0.45) MDM2RIPK1SLC16A3SLC16A1GPBAR1
SCHEMBL3703232 0.82 SLC16A3 (0.31) SLC16A3SLC16A1
SCHEMBL4566348 0.81 PTGER2 (0.33) RIPK1
SCHEMBL4194770 0.81

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2190822-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2010-06-02 EP disclosed
WO-2009041705-A9 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL (JP) 2009-08-13 WO disclosed
WO-2009041705-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-04-02 WO disclosed