SCHEMBL3700341

SCHEMBL3700341

CN(Cc1cc(Sc2cccc(Br)c2)n(-c2cc(F)ccc2F)n1)C(=O)OC(C)(C)C

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 8/20 0.44
SLC6A4 P31645 8/20 0.44
HTR2A P28223 1/20 0.44
CNR2 P34972 1/20 0.33
MAPT P10636 1/20 0.32
RIPK1 Q13546 2/20 0.31
IDH1 O75874 1/20 0.31
SOS1 Q07889 1/20 0.30
SLC16A3 O15427 1/20 0.30
SLC16A1 P53985 1/20 0.30
AAK1 Q2M2I8 1/20 0.30
HTT P42858 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4120953 0.88 MAPT (0.34) HTR2CSLC6A4HTR2ACNR2MAPT
SCHEMBL3692821 0.85 HTR2C (0.49) HTR2CSLC6A4HTR2ASLC16A3SLC16A1
SCHEMBL3699694 0.83 HTR2C (0.45) HTR2CSLC6A4HTR2ACNR2RIPK1
SCHEMBL3700345 0.82 MAPT (0.32) CNR2MAPT
SCHEMBL3805129 0.81 HTR2C (0.45) HTR2CSLC6A4HTR2AMAPT
SCHEMBL3690712 0.79 HTR2C (0.45) HTR2CSLC6A4HTR2ACNR2SLC16A3
SCHEMBL3693917 0.78 RIPK1 (0.32) MAPTRIPK1HTT
SCHEMBL3700342 0.77 RIPK1 (0.32) CNR2MAPTRIPK1
SCHEMBL4120959 0.76 MAPT (0.34) CNR2MAPTRIPK1
SCHEMBL3701837 0.76 HTR2C (0.43) HTR2CSLC6A4HTR2ACNR2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2190822-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2010-06-02 EP disclosed
WO-2009041705-A9 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL (JP) 2009-08-13 WO disclosed
WO-2009041705-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-04-02 WO disclosed