SCHEMBL3700345

SCHEMBL3700345

CC(C)(C)CN(Cc1cc(Sc2cccc(Br)c2)n(-c2cc(F)ccc2F)n1)C(=O)O

nearest known ligand 0.32

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.32
CNR2 P34972 1/20 0.32
TP53 P04637 1/20 0.32
ALDH1A1 P00352 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4120953 0.87 MAPT (0.34) MAPTCNR2ALDH1A1NPSR1
SCHEMBL3692824 0.84 SLC16A3 (0.36) MAPT
SCHEMBL3812505 0.82 CNR2 (0.33) CNR2
SCHEMBL3700341 0.82 HTR2C (0.44) MAPTCNR2
SCHEMBL3700342 0.79 RIPK1 (0.32) MAPTCNR2TP53ALDH1A1NPSR1
SCHEMBL4120959 0.79 MAPT (0.34) MAPTCNR2TP53ALDH1A1NPSR1
SCHEMBL3690717 0.78 ALDH1A1 (0.33) MAPTCNR2ALDH1A1NPSR1
SCHEMBL3693917 0.77 RIPK1 (0.32) MAPTALDH1A1NPSR1
SCHEMBL3706263 0.76 CNR2 (0.36) CNR2NPSR1
SCHEMBL3703723 0.76 KCNQ3 (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2190822-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2010-06-02 EP disclosed
WO-2009041705-A9 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL (JP) 2009-08-13 WO disclosed
WO-2009041705-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-04-02 WO disclosed