SCHEMBL3700342

SCHEMBL3700342

CC(C)(C)C(Cc1cc(Sc2cccc(Br)c2)n(-c2cc(F)ccc2F)n1)NC(=O)O

nearest known ligand 0.32

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
RIPK1 Q13546 1/20 0.32
MAPT P10636 3/20 0.32
ALDH1A1 P00352 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
CNR2 P34972 1/20 0.31
TP53 P04637 1/20 0.31
MAPK14 Q16539 1/20 0.30
NPY5R Q15761 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3692822 0.85 SLC16A3 (0.35) MAPTALDH1A1NPSR1
SCHEMBL3812496 0.83 KCNQ3 (0.33) RIPK1CNR2MAPK14
SCHEMBL4120959 0.82 MAPT (0.34) RIPK1MAPTALDH1A1NPSR1CNR2
SCHEMBL4120953 0.79 MAPT (0.34) RIPK1MAPTALDH1A1NPSR1CNR2
SCHEMBL3700345 0.79 MAPT (0.32) MAPTALDH1A1NPSR1CNR2TP53
SCHEMBL3690715 0.79 FPR1 (0.33) MAPTALDH1A1CNR2
SCHEMBL3693917 0.78 RIPK1 (0.32) RIPK1MAPTALDH1A1NPSR1MAPK14
SCHEMBL2836132 0.77 RIPK1 (0.36) RIPK1MAPTALDH1A1NPSR1CNR2
SCHEMBL3700341 0.77 HTR2C (0.44) RIPK1MAPTCNR2
SCHEMBL3695015 0.76 DHODH (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2190822-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2010-06-02 EP disclosed
WO-2009041705-A9 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL (JP) 2009-08-13 WO disclosed
WO-2009041705-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-04-02 WO disclosed