SCHEMBL3700575

SCHEMBL3700575

COc1cc(Sc2cc(CN(CC(C)(C)C)C(=O)O)nn2-c2ccccc2Cl)ccn1

nearest known ligand 0.40

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SLC16A3 O15427 14/20 0.40
SLC16A1 P53985 13/20 0.40
ALDH1A1 P00352 1/20 0.37
CTSA P10619 1/20 0.34
BRAF P15056 1/20 0.33
PDE4B Q07343 1/20 0.32
HTR2C P28335 1/20 0.32
SLC6A4 P31645 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4132125 0.88 SLC16A3 (0.40) SLC16A3SLC16A1ALDH1A1CTSAPDE4B
SCHEMBL3700571 0.84 HTR2C (0.47) SLC16A3SLC16A1ALDH1A1BRAFHTR2C
SCHEMBL3694441 0.84 SLC16A3 (0.40) SLC16A3SLC16A1BRAFPDE4BHTR2C
SCHEMBL3701902 0.84 SLC16A3 (0.38) SLC16A3SLC16A1PDE4BHTR2CSLC6A4
SCHEMBL3692824 0.84 SLC16A3 (0.36) SLC16A3SLC16A1BRAFPDE4BHTR2C
SCHEMBL3029606 0.84 SLC16A3 (0.38) SLC16A3SLC16A1PDE4BHTR2CSLC6A4
SCHEMBL3690040 0.82 SLC16A3 (0.34) SLC16A3SLC16A1
SCHEMBL3698141 0.81 SLC16A3 (0.37) SLC16A3SLC16A1PDE4B
SCHEMBL4132130 0.81 SLC16A3 (0.38) SLC16A3SLC16A1ALDH1A1CTSAPDE4B
SCHEMBL3700573 0.80 SLC16A3 (0.39) SLC16A3SLC16A1ALDH1A1CTSABRAF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2190822-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2010-06-02 EP disclosed
WO-2009041705-A9 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL (JP) 2009-08-13 WO disclosed
WO-2009041705-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-04-02 WO disclosed