SCHEMBL3700573

SCHEMBL3700573

COc1cc(Sc2cc(CC(NC(=O)O)C(C)(C)C)nn2-c2ccccc2Cl)ccn1

nearest known ligand 0.39

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SLC16A3 O15427 10/20 0.39
SLC16A1 P53985 9/20 0.39
CTSA P10619 3/20 0.38
ALDH1A1 P00352 1/20 0.34
BRAF P15056 1/20 0.34
ADORA1 P30542 1/20 0.32
CNR1 P21554 2/20 0.32
CCKAR P32238 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3694436 0.85 SLC16A3 (0.39) SLC16A3SLC16A1CTSABRAF
SCHEMBL3029599 0.83 SLC16A3 (0.37) SLC16A3SLC16A1ALDH1A1CNR1
SCHEMBL3701900 0.83 SLC16A3 (0.37) SLC16A3SLC16A1ALDH1A1CNR1
SCHEMBL3692822 0.83 SLC16A3 (0.35) SLC16A3SLC16A1ALDH1A1BRAFCNR1
SCHEMBL4132130 0.83 SLC16A3 (0.38) SLC16A3SLC16A1CTSAALDH1A1ADORA1
SCHEMBL3698138 0.82 SLC16A3 (0.38) SLC16A3SLC16A1ALDH1A1CNR1
SCHEMBL3700575 0.80 SLC16A3 (0.40) SLC16A3SLC16A1CTSAALDH1A1BRAF
SCHEMBL4132125 0.80 SLC16A3 (0.40) SLC16A3SLC16A1CTSAALDH1A1CNR1
SCHEMBL3698799 0.79 SLC16A3 (0.40) SLC16A3SLC16A1CTSAALDH1A1BRAF
SCHEMBL4201749 0.79 SLC16A3 (0.36) SLC16A3SLC16A1CTSACNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2190822-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2010-06-02 EP disclosed
WO-2009041705-A9 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL (JP) 2009-08-13 WO disclosed
WO-2009041705-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-04-02 WO disclosed