SCHEMBL3700700

SCHEMBL3700700

Cc1ccc(S(=O)(=O)c2cc(CN(C)C(=O)OC(C)(C)C)nn2-c2cccc(F)c2C)cn1

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 8/20 0.38
SLC6A4 P31645 8/20 0.38
HTR2A P28223 1/20 0.38
RXRA P19793 2/20 0.33
GRIN1 Q05586 2/20 0.33
GRIN2B Q13224 2/20 0.33
NAMPT P43490 1/20 0.32
SCN9A Q15858 4/20 0.31
SCN5A Q14524 1/20 0.31
SLC16A3 O15427 2/20 0.31
SLC16A1 P53985 2/20 0.31
ATM Q13315 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
F2 P00734 1/20 0.31
CACNA1G O43497 1/20 0.30
CACNA1B Q00975 1/20 0.30
CACNA1C Q13936 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3703100 0.95 HTR2C (0.36) HTR2CSLC6A4HTR2ARXRAGRIN1
SCHEMBL3700608 0.94 HTR2C (0.40) HTR2CSLC6A4HTR2ANAMPTSCN9A
SCHEMBL3697673 0.92 HTR2C (0.39) HTR2CSLC6A4HTR2ARXRAGRIN1
SCHEMBL3699812 0.90 HTR2C (0.38) HTR2CSLC6A4HTR2ARXRAGRIN1
SCHEMBL3688570 0.90 HTR2C (0.38) HTR2CSLC6A4HTR2ARXRAGRIN1
SCHEMBL3698341 0.89 HTR2C (0.38) HTR2CSLC6A4HTR2ANAMPTF2
SCHEMBL4125819 0.88 PTGS2 (0.33) HTR2CHTR2ARXRAGRIN1GRIN2B
SCHEMBL3696612 0.88 HTR2C (0.42) HTR2CSLC6A4HTR2ASLC16A3SLC16A1
SCHEMBL4200021 0.88 HTR2C (0.36) HTR2CSLC6A4HTR2ASLC16A3SLC16A1
SCHEMBL3697102 0.85 HTR2C (0.41) HTR2CSLC6A4HTR2ANAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2190822-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2010-06-02 EP disclosed
WO-2009041705-A9 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL (JP) 2009-08-13 WO disclosed
WO-2009041705-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-04-02 WO disclosed