SCHEMBL3697102

SCHEMBL3697102

Cc1ccc(S(=O)(=O)c2cc(CN(C)C(=O)OC(C)(C)C)nn2-c2cc(F)ccc2Cl)cn1

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 9/20 0.41
SLC6A4 P31645 8/20 0.41
HTR2A P28223 2/20 0.41
KAT6A Q92794 2/20 0.33
KAT5 Q92993 2/20 0.33
PRCP P42785 2/20 0.32
P2RX7 Q99572 1/20 0.32
NAMPT P43490 1/20 0.31
KAT8 Q9H7Z6 1/20 0.31
NR1I2 O75469 1/20 0.31
KCNH2 Q12809 1/20 0.30
GPBAR1 Q8TDU6 1/20 0.30
GPR6 P46095 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3696612 0.90 HTR2C (0.42) HTR2CSLC6A4HTR2A
SCHEMBL3705293 0.89 HTR2C (0.39) HTR2CSLC6A4HTR2ANAMPT
SCHEMBL3704890 0.88 P2RX7 (0.34) HTR2CHTR2APRCPP2RX7NAMPT
SCHEMBL3688570 0.88 HTR2C (0.38) HTR2CSLC6A4HTR2AKAT6AKAT5
SCHEMBL3703585 0.87 HTR2C (0.41) HTR2CSLC6A4HTR2AKAT6AKAT5
SCHEMBL3706785 0.87 HTR2C (0.40) HTR2CSLC6A4HTR2AGPR6
SCHEMBL3700978 0.86 HTR2C (0.45) HTR2CSLC6A4HTR2AKAT6AKAT5
SCHEMBL3700608 0.86 HTR2C (0.40) HTR2CSLC6A4HTR2ANAMPTKCNH2
SCHEMBL3698341 0.85 HTR2C (0.38) HTR2CSLC6A4HTR2ANAMPT
SCHEMBL3700700 0.85 HTR2C (0.38) HTR2CSLC6A4HTR2ANAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2190822-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2010-06-02 EP disclosed
WO-2009041705-A9 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL (JP) 2009-08-13 WO disclosed
WO-2009041705-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-04-02 WO disclosed