SCHEMBL3700852

SCHEMBL3700852

CC(C)(C)C(Cc1cc(S(=O)(=O)c2cccnc2)n(-c2cc(F)ccc2Cl)n1)NC(=O)O.CC(C)(C)C(Cc1cc(Sc2cccnc2)n(-c2cc(F)ccc2Cl)n1)NC(=O)O

nearest known ligand 0.36

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
FPR1 P21462 1/20 0.36
NAMPT P43490 1/20 0.31
ABCC9 O60706 1/20 0.30
ABCC8 Q09428 1/20 0.30
KCNJ11 Q14654 1/20 0.30
KCNJ8 Q15842 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3705290 0.92 FPR1 (0.41) FPR1NAMPTABCC9ABCC8KCNJ11
SCHEMBL3690715 0.92 FPR1 (0.33) FPR1
SCHEMBL3706679 0.91 FPR1 (0.33) FPR1ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL3693159 0.85 FPR1 (0.42) FPR1NAMPTABCC9ABCC8KCNJ11
SCHEMBL3700854 0.83 NAMPT (0.30) NAMPT
SCHEMBL3701900 0.82 SLC16A3 (0.37)
SCHEMBL4566346 0.82 FPR1 (0.38) FPR1NAMPTABCC9ABCC8KCNJ11
SCHEMBL3702435 0.81 RIPK1 (0.36) FPR1
SCHEMBL3700851 0.81 HTR2C (0.39)
SCHEMBL3703720 0.80 KCNQ3 (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2190822-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2010-06-02 EP disclosed
WO-2009041705-A9 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL (JP) 2009-08-13 WO disclosed
WO-2009041705-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-04-02 WO disclosed