SCHEMBL3700876

SCHEMBL3700876

N#Cc1ccc2c(c1)CC=NO2

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PNMT P11086 6/20 0.38
DRD2 P14416 2/20 0.38
DRD3 P35462 2/20 0.38
CA12 O43570 1/20 0.34
CA9 Q16790 1/20 0.34
CYP2A6 P11509 1/20 0.33
USP2 O75604 1/20 0.32
TRPA1 O75762 1/20 0.32
CYP11B1 P15538 1/20 0.31
CYP11B2 P19099 1/20 0.31
KDM1A O60341 1/20 0.31
HTR2A P28223 1/20 0.31
HTR2C P28335 1/20 0.31
HTR2B P41595 1/20 0.31
CYP19A1 P11511 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6253306 0.73 AHR (0.39) PNMT
SCHEMBL8612336 0.70 PNMT (0.39) PNMTDRD2DRD3CA12CA9
SCHEMBL11017385 0.69 TRPA1 (0.44) PNMTDRD2DRD3TRPA1CYP11B1
SCHEMBL4967364 0.68 DRD2 (0.47) PNMTDRD2DRD3CA12CA9
SCHEMBL3523194 0.66 PNMT (0.41) PNMTDRD2DRD3CA12CA9
SCHEMBL3492241 0.66 PRKCI (0.47) PNMTDRD2DRD3
SCHEMBL7038650 0.66 TRPA1 (0.44) PNMTDRD2DRD3TRPA1CYP11B1
SCHEMBL28664612 0.64 CA12 (0.46) CA12CA9CYP2A6USP2TRPA1
SCHEMBL1786744 0.63 PNMT (0.50) PNMTDRD2DRD3CA12CA9
SCHEMBL28482571 0.63 PNMT (0.42) PNMTDRD2DRD3CA12CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2748157-A1 METHOD FOR PRODUCING TETRAZOLE-SUBSTITUTED ANTHRANILIC ACID DIAMIDE DERIVATIVES BY REACTING BENZOXAZINONES WITH AMINES Bayer Intellectual Property GmbH (DE) 2014-07-02 EP disclosed
WO-2013030100-A1 METHOD FOR PRODUCING TETRAZOLE-SUBSTITUTED ANTHRANILIC ACID DIAMIDE DERIVATIVES BY REACTING BENZOXAZINONES WITH AMINES BAYER INTELLECTUAL PROPERTY GMBH (DE) 2013-03-07 WO disclosed
EP-2203459-A1 SPIROCYCLIC AMINOQUINOLONES AS GSK-3 INHIBITORS Activx Biosciences, Inc. (US) 2010-07-07 EP disclosed
WO-2009035684-A1 SPIROCYCLIC AMINOQUINOLONES AS GSK-3 INHIBITORS ACTIVX BIOSCIENCES, INC. (US) 2009-03-19 WO disclosed