SCHEMBL1728006

SCHEMBL1728006

O=C(O)NC(c1cc(-n2ccnc2)ncn1)C1CCNCC1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P4HTM Q9NXG6 1/20 0.37
CYP1A2 P05177 5/20 0.36
CYP3A4 P08684 5/20 0.36
CYP2D6 P10635 4/20 0.36
ALOX15 P16050 4/20 0.36
HSD17B10 Q99714 4/20 0.36
CLK4 Q9HAZ1 3/20 0.36
CYP2C19 P33261 4/20 0.36
TSHR P16473 1/20 0.36
LMNA P02545 2/20 0.35
MAPT P10636 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
SMYD3 Q9H7B4 3/20 0.35
AKT1 P31749 2/20 0.35
CDK2 P24941 1/20 0.35
CHRNA7 P36544 2/20 0.35
HTR3A P46098 2/20 0.35
EGLN2 Q96KS0 1/20 0.34
TLR9 Q9NR96 1/20 0.34
TLR8 Q9NR97 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3701313 0.75 AKT1 (0.43) SMYD3AKT1CDK2
SCHEMBL1729045 0.73 F11 (0.45) SMYD3AKT1CDK2
SCHEMBL18431062 0.69 CYP3A4 (0.48) CYP1A2CYP3A4CYP2D6ALOX15HSD17B10
SCHEMBL27600626 0.66 AKT1 (0.41) SMYD3AKT1CDK2
SCHEMBL17250004 0.66 CYP3A4 (0.50) CYP1A2CYP3A4CYP2D6ALOX15HSD17B10
SCHEMBL25135722 0.65 CD38 (0.49) CYP2D6CYP2C19SMYD3
SCHEMBL30363752 0.65 CD38 (0.49) CYP2D6CYP2C19SMYD3
SCHEMBL13472422 0.65 CYP1A2 (0.50) P4HTMCYP1A2CYP3A4CYP2D6ALOX15
SCHEMBL1727781 0.65 SMYD3 (0.43) SMYD3AKT1CDK2
SCHEMBL9521235 0.65 CYP3A4 (0.58) CYP1A2CYP3A4CYP2D6ALOX15HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1633735-B1 DERIVATIVES OF PIPERIDINYL- AND PIPERAZINYL-ALKYL CARBAMATES, PREPARATION METHODS THEREOF AND APPLICATION OF SAME IN THERAPEUTICS SANOFI SA (FR) 2011-11-30 EP claimed