SCHEMBL3702935

SCHEMBL3702935

COC([O])C(=O)c1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.50
TDP1 Q9NUW8 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
ALDH1A1 P00352 4/20 0.47
CYP3A4 P08684 1/20 0.47
CES2 O00748 3/20 0.47
CES1 P23141 3/20 0.47
LMNA P02545 3/20 0.47
PGR P06401 1/20 0.44
ADRA2A P08913 1/20 0.44
ADRA2B P18089 1/20 0.44
HTR2A P28223 1/20 0.44
HRH1 P35367 1/20 0.44
KCNH2 Q12809 1/20 0.44
HTT P42858 2/20 0.44
MDM2 Q00987 1/20 0.44
KMT2A Q03164 3/20 0.43
F2 P00734 1/20 0.43
NPC1 O15118 3/20 0.42
MAPT P10636 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL316378 0.81 TSHR (0.48) TSHRTDP1L3MBTL1ALDH1A1CYP3A4
Benzene SCHEMBL27641543 0.80 TSHR (0.52) TSHRTDP1L3MBTL1ALDH1A1CYP3A4
SCHEMBL26712 0.80 TSHR (0.52) TSHRTDP1L3MBTL1ALDH1A1CYP3A4
SCHEMBL146504 0.80 TSHR (0.52) TSHRTDP1L3MBTL1ALDH1A1CYP3A4
SCHEMBL28197933 0.80 TSHR (0.52) TSHRTDP1L3MBTL1ALDH1A1CYP3A4
SCHEMBL5245130 0.78 CES2 (0.52) TSHRTDP1L3MBTL1ALDH1A1CYP3A4
SCHEMBL34992 0.78 CES2 (0.52) TSHRTDP1L3MBTL1ALDH1A1CYP3A4
SCHEMBL2598221 0.78 MAPT (0.53) TSHRTDP1L3MBTL1ALDH1A1CYP3A4
SCHEMBL2231539 0.77 TSHR (0.48) TSHRTDP1L3MBTL1ALDH1A1CYP3A4
SCHEMBL4303850 0.77 TSHR (0.48) TSHRTDP1L3MBTL1ALDH1A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0123441-B1 VINCALEUKOBLASTINE DERIVATIVES LILLY INDUSTRIES LIMITED (GB) 1990-10-03 EP claimed
US-4675400-A FORM CONJUGATES WITH IMMUNOGLOBULINS; ANTITUMOR AGENTS ELI LILLY AND COMPANY (US) 1987-06-23 US claimed
US-4596676-A Bifunctional ester derivatives of 4-desacetyl indole-dihydroindole alkaloids LILLY INDUSTRIES LIMITED (GB) 1986-06-24 US claimed
EP-0123441-A1 Vincaleukoblastine derivatives LILLY INDUSTRIES LIMITED (GB) 1984-10-31 EP claimed
EP-2396017-A1 APOLIPOPROTEIN A-I MIMICS Cerenis Therapeutics SA (FR) 2011-12-21 EP disclosed
WO-2010093918-A1 APOLIPOPROTEIN A-I MIMICS CERENIS THERAPEUTICS SA (FR) 2010-08-19 WO disclosed
EP-0123441-B1 VINCALEUKOBLASTINE DERIVATIVES LILLY INDUSTRIES LIMITED (GB) 1990-10-03 EP disclosed
US-4675400-A FORM CONJUGATES WITH IMMUNOGLOBULINS; ANTITUMOR AGENTS ELI LILLY AND COMPANY (US) 1987-06-23 US disclosed
US-4596676-A Bifunctional ester derivatives of 4-desacetyl indole-dihydroindole alkaloids LILLY INDUSTRIES LIMITED (GB) 1986-06-24 US disclosed
EP-0123441-A1 Vincaleukoblastine derivatives LILLY INDUSTRIES LIMITED (GB) 1984-10-31 EP disclosed