Bicarbonate

Bicarbonate

SCHEMBL3704738

C[C@@H]([C@@H](C(=O)Nc1cccc(CC2CC2)c1)c1ccc(CN2Cc3ccccc3C2=O)cc1)C(F)(F)F.O=C(O)O

nearest known ligand 0.45

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

GSK3AGSK3BIMPA1

The experimentally established mechanism targets of Bicarbonate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.41
THRB P10828 3/20 0.40
MAPT P10636 4/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
HDAC1 Q13547 2/20 0.39
HDAC7 Q8WUI4 1/20 0.39
LMNA P02545 1/20 0.39
ACKR3 P25106 2/20 0.39
CCR3 P51677 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bicarbonate SCHEMBL3702662 1.00 ACHE (0.41) ACHETHRBMAPTMEN1KMT2A
Bicarbonate SCHEMBL3696349 0.89 ACKR3 (0.36) THRBACKR3CCR3
Bicarbonate SCHEMBL3698645 0.89 ACKR3 (0.36) THRBACKR3CCR3
SCHEMBL13660768 0.88 THRB (0.40) THRBMAPTMEN1KMT2AHDAC1
SCHEMBL3704735 0.88 THRB (0.40) THRBMAPTMEN1KMT2AHDAC1
SCHEMBL3702660 0.88 THRB (0.40) THRBMAPTMEN1KMT2AHDAC1
SCHEMBL3696153 0.86 MEN1 (0.42) THRBMAPTMEN1KMT2AHDAC1
SCHEMBL7602101 0.86 MAPT (0.40) THRBMAPTMEN1KMT2AHDAC1
SCHEMBL7606170 0.86 MAPT (0.40) THRBMAPTMEN1KMT2AHDAC1
Bicarbonate SCHEMBL3697242 0.83 MAPT (0.46) ACHETHRBMAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2268625-B1 OXO-HETEROCYCLIC SUBSTITUTED CARBOXYLIC ACID DERIVATES AND THE USE THEREOF Bayer Pharma AG (DE) 2012-05-16 EP disclosed