Cefoperazone

Cefoperazone

SCHEMBL37056

CCN1CCN(C(=O)N[C@@H](C(=O)N[C@@H]2C(=O)N3C(C(=O)O)=C(CSc4nnnn4C)CS[C@H]23)c2ccc(O)cc2)C(=O)C1=O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

dacAdacBdacCftsImrcAmrcBmrdA

The experimentally established mechanism targets of Cefoperazone. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 10/20 1.00
SLC22A6 Q4U2R8 2/20 1.00
SLC22A8 Q8TCC7 2/20 1.00
SLC22A11 Q9NSA0 2/20 1.00
PDE3A Q14432 1/20 1.00
HSD17B10 Q99714 4/20 0.99
THRB P10828 1/20 0.99
TSHR P16473 1/20 0.99
TDP1 Q9NUW8 10/20 0.88
NR1I2 O75469 2/20 0.62
PGR P06401 2/20 0.62
PPARG P37231 1/20 0.62
POLB P06746 10/20 0.56
ALDH1A1 P00352 5/20 0.56
HTT P42858 1/20 0.56
KDM4E B2RXH2 1/20 0.55
CYP3A4 P08684 1/20 0.55
HPGD P15428 1/20 0.55
APEX1 P27695 1/20 0.55
PTPN7 P35236 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Cefoperazone SCHEMBL9326569 1.00 MAPT (1.00) MAPTSLC22A6SLC22A8SLC22A11PDE3A
Cefoperazone SCHEMBL16091123 1.00 MAPT (1.00) MAPTSLC22A6SLC22A8SLC22A11PDE3A
Cefoperazone SCHEMBL11522109 1.00 MAPT (1.00) MAPTSLC22A6SLC22A8SLC22A11PDE3A
Cefoperazone SCHEMBL2222952 1.00 MAPT (1.00) MAPTSLC22A6SLC22A8SLC22A11PDE3A
Cefoperazone SCHEMBL18061225 1.00 MAPT (1.00) MAPTSLC22A6SLC22A8SLC22A11PDE3A
Cefoperazone SCHEMBL16072819 1.00 MAPT (1.00) MAPTSLC22A6SLC22A8SLC22A11PDE3A
Cefoperazone SCHEMBL15387468 1.00 MAPT (1.00) MAPTSLC22A6SLC22A8SLC22A11PDE3A
Cefoperazone SCHEMBL3758644 0.99 HSD17B10 (1.00) MAPTSLC22A6SLC22A8SLC22A11PDE3A
Cefoperazone SCHEMBL40452 0.99 MAPT (0.99) MAPTSLC22A6SLC22A8SLC22A11PDE3A
Cefoperazone SCHEMBL28649126 0.99 MAPT (0.99) MAPTSLC22A6SLC22A8SLC22A11PDE3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 26136 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4747395-A1 A KIT FOR IDENTIFYING BACTERIA AND DETERMINING ANTIBIOTIC SENSITIVITY Diagopreutic Private Limited (IN) 2026-05-27 EP claimed
US-12637481-B2 Boronic acid derivatives and therapeutic uses thereof QPEX BIOPHARMA, INC. (US) 2026-05-26 US claimed
CN-122071712-A Beta-lactam antibiotic whole-cell biosensor, construction method and application 中国科学院天津工业生物技术研究所 2026-05-22 CN claimed
CN-122035989-A Method for reducing runoff pollution load of river bank zone 中国长江三峡集团有限公司 2026-05-15 CN claimed
US-12622919-B2 Methods for treating hypervirulent Klebsiella pneumoniae infection CITY UNIVERSITY OF HONG KONG (CN) 2026-05-12 US claimed
US-20260108619-A1 CONJUGATION LINKERS, CELL BINDING MOLECULE-DRUG CONJUGATES CONTAINING THE LINKERS, METHODS OF MAKING AND USES SUCH CONJUGATES WITH THE LINKERS HANGZHOU DAC BIOTECH CO., LTD. (CN) 2026-04-23 US claimed
EP-4725496-A2 N-[4-[1-(1,4-DIOXASPIRO[4.5]DEC-8-YL)-4-(8-OXA-3-AZABICYCLO[3.2.1]OCT-3-YL)-1H-PYRAZOLO[3,4-D]PYRIMIDIN-6-YL]PHENYL]-N'-METHYLUREA FOR USE IN THE TREATMENT OF COVID19 NantCell, Inc. (US) 2026-04-15 EP claimed
US-12590108-B2 Boracic acid compound PHAENO THERAPEUTICS CO., LTD (CN) 2026-03-31 US claimed
US-12576124-B2 Formulation of a conjugate of a tubulysin analog to a cell-binding molecule HANGZHOU DAC BIOTECH CO., LTD (CN) 2026-03-17 US claimed
US-20260034183-A1 TREATMENT OF CLOSTRIDIUM DIFFICILE INFECTION VEDANTA BIOSCIENCES, INC. (US) 2026-02-05 US claimed
US-4503040-A 6-(Aminoacyloxymethyl)penicillanic acid 1,1-dioxides as beta-lactamase inhibitors PFIZER INC. (US) 1985-03-05 US claimed
EP-0118196-A1 Process for the manufacture of highly crystalline sodium cefoperazone PFIZER INC. (US) 1984-09-12 EP claimed
US-4458070-A Process for the manufacture of crystalline sodium cefoperazone PFIZER INC. (US) 1984-07-03 US claimed
US-4456753-A Process for the manufacture of highly crystalline sodium cefoperazone PFIZER INC. (US) 1984-06-26 US claimed
US-4452796-A ANTIBIOTICS PFIZER INC. (US) 1984-06-05 US claimed
EP-0101170-A1 Process for the manufacture of sodium cefoperazone PFIZER INC. (US) 1984-02-22 EP claimed
US-4427678-A 6-Aminomethylpenicillanic acid 1,1-dioxide derivatives as beta-lactamase inhibitors PFIZER INC. (US) 1984-01-24 US claimed
EP-0084925-A1 6-Aminoalkylpenicillanic acid 1,1-dioxides and derivatives as beta-lactamase inhibitors PFIZER INC. (US) 1983-08-03 EP claimed
WO-1982003090-A1 METHOD AND KIT FOR IDENTIFICATION OF BETA-LACTAMASES JAMES RICHARD 1982-09-16 WO claimed
EP-0059645-A1 Method and kit for identification of beta-lactamases NATIONAL RESEARCH DEVELOPMENT CORPORATION (GB) 1982-09-08 EP claimed