Cefoperazone

Cefoperazone

SCHEMBL40452

CCN1CCN(C(=O)N[C@@H](C(=O)N[C@@H]2C(=O)N3C(C(=O)O)=C(CSc4nnnn4C)CS[C@H]23)c2ccc(O)cc2)C(=O)C1=O.[NaH]

nearest known ligand 0.99

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

dacAdacBdacCftsImrcAmrcBmrdA

The experimentally established mechanism targets of Cefoperazone. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 10/20 0.99
SLC22A6 Q4U2R8 2/20 0.99
SLC22A8 Q8TCC7 2/20 0.99
SLC22A11 Q9NSA0 2/20 0.99
PDE3A Q14432 1/20 0.99
HSD17B10 Q99714 4/20 0.98
THRB P10828 1/20 0.98
TSHR P16473 1/20 0.98
TDP1 Q9NUW8 10/20 0.87
NR1I2 O75469 2/20 0.62
PGR P06401 2/20 0.62
PPARG P37231 1/20 0.62
POLB P06746 10/20 0.56
ALDH1A1 P00352 5/20 0.56
HTT P42858 1/20 0.55
KDM4E B2RXH2 1/20 0.55
CYP3A4 P08684 1/20 0.55
HPGD P15428 1/20 0.55
APEX1 P27695 1/20 0.55
PTPN7 P35236 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Cefoperazone SCHEMBL27651465 1.00 MAPT (0.99) MAPTSLC22A6SLC22A8SLC22A11PDE3A
Cefoperazone SCHEMBL16091123 0.99 MAPT (1.00) MAPTSLC22A6SLC22A8SLC22A11PDE3A
Cefoperazone SCHEMBL37056 0.99 MAPT (1.00) MAPTSLC22A6SLC22A8SLC22A11PDE3A
Cefoperazone SCHEMBL11522109 0.99 MAPT (1.00) MAPTSLC22A6SLC22A8SLC22A11PDE3A
Cefoperazone SCHEMBL2222952 0.99 MAPT (1.00) MAPTSLC22A6SLC22A8SLC22A11PDE3A
Cefoperazone SCHEMBL16072819 0.99 MAPT (1.00) MAPTSLC22A6SLC22A8SLC22A11PDE3A
Cefoperazone SCHEMBL9326569 0.99 MAPT (1.00) MAPTSLC22A6SLC22A8SLC22A11PDE3A
Cefoperazone SCHEMBL18061225 0.99 MAPT (1.00) MAPTSLC22A6SLC22A8SLC22A11PDE3A
Cefoperazone SCHEMBL15387468 0.99 MAPT (1.00) MAPTSLC22A6SLC22A8SLC22A11PDE3A
Cefoperazone SCHEMBL3758644 0.99 HSD17B10 (1.00) MAPTSLC22A6SLC22A8SLC22A11PDE3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 4233 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117482095-B Cefoperazone sodium and sulbactam sodium composition and preparation method thereof CHENGDU JINGFU PHARMACEUTICAL TECHNOLOGY Co.,Ltd. (CN) 2026-05-26 CN claimed
WO-2025111413-A1 TREATMENT FOR SKIN DISORDERS Mycotechnology, Inc. (US) 2025-05-30 WO claimed
CN-119818504-A Antibacterial composition of cefoperazone and avibactam and application thereof 重庆圣华曦药业股份有限公司 2025-04-15 CN claimed
US-12274830-B2 Nitric oxide inhalation therapy for infants with bronchiolitis BEYOND AIR LTD (IL) 2025-04-15 US claimed
CN-119391643-B Culture medium and method for culturing digestive tract tumor by using three-dimensional tumor tablet technology 珠海澳大科技研究院 2025-03-14 CN claimed
CN-115684393-B Two-dimensional detection method for impurities in cefoperazone sodium and sulbactam sodium for injection 北京悦康科创医药科技股份有限公司 2025-02-25 CN claimed
CN-119438454-A Cefoperazone sodium sulbactam sodium polymer for injection and specific impurity analysis method 哈药集团技术中心 2025-02-14 CN claimed
CN-119438417-A Method for detecting polymer in cefoperazone sodium and sulbactam sodium 海南卫康制药(潜山)有限公司 2025-02-14 CN claimed
CN-119391643-A Culture medium and method for culturing digestive tract tumor by using three-dimensional tumor tablet technology 珠海澳大科技研究院 2025-02-07 CN claimed
CN-222117262-U Sealed filling mechanism of cefoperazone sodium and sulbactam sodium 山西振东泰盛制药有限公司 2024-12-06 CN claimed
WO-2002030469-A2 BETA-LACTAM ANTIBIOTIC-POLYSACCHARIDE COMPLEX ORCHID CHEMICALS AND PHARMACEUTICALS LIMITED (IN) 2002-04-18 WO claimed
WO-2001079210-A2 A PROCESS FOR THE PREPARATION OF HIGHLY CRYSTALLINE SODIUM CEFOPERAZONE ANTIBIOTICOS S.P.A. (IT) 2001-10-25 WO claimed
US-6245735-B1 CONJUGATE OF ANTIBIOTIC AND POLYPEPTIDE OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR OR LIPOPOLYSACCHARIDE BINDING FRAGMENT THE BRIGHAM AND WOMEN'S HOSPITAL, INC. 2001-06-12 US claimed
US-4678512-A Marine coating compositions and method GRAMS RALPH R 1987-07-07 US claimed
EP-0118196-B1 PROCESS FOR THE MANUFACTURE OF HIGHLY CRYSTALLINE SODIUM CEFOPERAZONE PFIZER INC. (US) 1986-12-30 EP claimed
EP-0101170-B1 PROCESS FOR THE MANUFACTURE OF SODIUM CEFOPERAZONE PFIZER INC. (US) 1986-01-15 EP claimed
EP-0118196-A1 Process for the manufacture of highly crystalline sodium cefoperazone PFIZER INC. (US) 1984-09-12 EP claimed
US-4458070-A Process for the manufacture of crystalline sodium cefoperazone PFIZER INC. (US) 1984-07-03 US claimed
US-4456753-A Process for the manufacture of highly crystalline sodium cefoperazone PFIZER INC. (US) 1984-06-26 US claimed
EP-0101170-A1 Process for the manufacture of sodium cefoperazone PFIZER INC. (US) 1984-02-22 EP claimed