SCHEMBL3706785

SCHEMBL3706785

CN(Cc1cc(S(=O)(=O)c2ccc(Cl)nc2)n(-c2ccc(F)cc2F)n1)C(=O)OC(C)(C)C.Cc1ccc(S(=O)(=O)c2cc(CN(C)C(=O)O)nn2-c2ccc(F)cc2F)cn1

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 8/20 0.40
SLC6A4 P31645 8/20 0.40
HTR2A P28223 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.32
CNR2 P34972 4/20 0.32
CNR1 P21554 2/20 0.32
ALDH1A1 P00352 2/20 0.32
THRB P10828 1/20 0.32
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
LMNA P02545 1/20 0.31
TP53 P04637 1/20 0.31
KCNQ3 O43525 1/20 0.30
KCNQ2 O43526 1/20 0.30
GPR6 P46095 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4200021 0.90 HTR2C (0.36) HTR2CSLC6A4HTR2AALDH1A1MEN1
SCHEMBL4130737 0.89 ALDH1A1 (0.38) HTR2CHTR2ASMN1; SMN2CNR2CNR1
SCHEMBL3706787 0.89 CNR1 (0.32) CNR2CNR1ALDH1A1THRBMEN1
SCHEMBL3700225 0.88 HTR2C (0.39) HTR2CSLC6A4HTR2AALDH1A1MEN1
SCHEMBL3698449 0.88 NR2F2 (0.35) HTR2CSLC6A4HTR2ACNR2CNR1
SCHEMBL3700978 0.87 HTR2C (0.45) HTR2CSLC6A4HTR2ACNR2ALDH1A1
SCHEMBL3703585 0.87 HTR2C (0.41) HTR2CSLC6A4HTR2AALDH1A1THRB
SCHEMBL3697102 0.87 HTR2C (0.41) HTR2CSLC6A4HTR2AGPR6
SCHEMBL3698341 0.87 HTR2C (0.38) HTR2CSLC6A4HTR2ATHRBLMNA
SCHEMBL3698587 0.85 HTR2C (0.42) HTR2CSLC6A4HTR2ASMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2190822-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2010-06-02 EP disclosed
WO-2009041705-A9 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL (JP) 2009-08-13 WO disclosed
WO-2009041705-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-04-02 WO disclosed