SCHEMBL3708930

SCHEMBL3708930

CCOC(=O)C(OC(=O)c1ccc2[nH]ccc2c1)C(C)=O

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 2/20 0.51
TAS1R3 Q7RTX0 1/20 0.46
TAS1R1 Q7RTX1 1/20 0.46
MAPT P10636 2/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2C19 P33261 1/20 0.45
RAB9A P51151 1/20 0.45
CTNNB1 P35222 3/20 0.44
WNT3A P56704 3/20 0.44
TUBB4A P04350 1/20 0.43
TUBB P07437 1/20 0.43
TUBA3C P0DPH7 1/20 0.43
TUBA1B P68363 1/20 0.43
TUBA4A P68366 1/20 0.43
TUBB4B P68371 1/20 0.43
TUBB3 Q13509 1/20 0.43
TUBB2A Q13885 1/20 0.43
TUBB8 Q3ZCM7 1/20 0.43
TUBA3E Q6PEY2 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1222893 0.84 MAOA (0.67) MAOATAS1R3TAS1R1MAPTCYP1A2
SCHEMBL31094660 0.84 MAOA (0.67) MAOATAS1R3TAS1R1MAPTCYP1A2
Hydrochloric Acid SCHEMBL28263903 0.83 MAOA (0.65) MAOATAS1R3TAS1R1MAPTCYP1A2
SCHEMBL6874059 0.81 MAOA (0.50) MAOATAS1R3TAS1R1MAPTCYP1A2
SCHEMBL1675118 0.78 CA12 (0.53) MAOATAS1R3TAS1R1MAPTCYP1A2
SCHEMBL27752787 0.76 TAS1R3 (0.50) MAOATAS1R3TAS1R1MAPTCYP1A2
SCHEMBL7493251 0.76 TAS1R3 (0.46) MAOATAS1R3TAS1R1MAPTCYP1A2
SCHEMBL8132038 0.75 TAS1R3 (0.57) MAOATAS1R3TAS1R1MAPTCYP1A2
SCHEMBL27752783 0.75 CTNNB1 (0.49) MAOATAS1R3TAS1R1MAPTCYP1A2
SCHEMBL9034535 0.74 MAOA (0.50) MAOATAS1R3TAS1R1MAPTCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010093191-A2 NOVEL COMPOUNDS EFFECTIVE AS XANTHINE OXIDASE INHIBITORS, METHOD FOR PREPARING THE SAME, AND PHARMACEUTICAL COMPOSITION CONTAINING THE SAME LG LIFE SCIENCES LTD. (KR) 2010-08-19 WO disclosed
WO-2010093191-A2 NOVEL COMPOUNDS EFFECTIVE AS XANTHINE OXIDASE INHIBITORS, METHOD FOR PREPARING THE SAME, AND PHARMACEUTICAL COMPOSITION CONTAINING THE SAME LG LIFE SCIENCES LTD. (KR) 2010-08-19 WO disclosed