SCHEMBL3709922

SCHEMBL3709922

CCOc1ccc(CN2CCN(C(=O)c3cc4cc(Oc5cc(C)c(NC(=O)c6ccc(Cl)c(Cl)c6)cn5)ccc4n3C)CC2)cc1

nearest known ligand 0.46

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 2/20 0.46
PRKAA2 P54646 2/20 0.46
STAT3 P40763 18/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL3065325 0.99 PIK3CA (0.46) PIK3CAPRKAA2STAT3
Bromide SCHEMBL3053365 0.89 PRKAA2 (0.47) PIK3CAPRKAA2STAT3
Oxalic Acid SCHEMBL3060675 0.88 PIK3CA (0.42) PIK3CAPRKAA2STAT3
SCHEMBL3052158 0.86 SMN1; SMN2 (0.46) PIK3CAPRKAA2STAT3
SCHEMBL3052627 0.86 LGALS8 (0.41) STAT3
Bromide SCHEMBL3061338 0.85 PIK3CA (0.45) PIK3CAPRKAA2STAT3
SCHEMBL3055575 0.85 HRH3 (0.41) PIK3CASTAT3
Bromide SCHEMBL3068012 0.83 PRKAA2 (0.46) PIK3CAPRKAA2STAT3
Bromide SCHEMBL3067536 0.83 FAAH (0.44) PIK3CAPRKAA2STAT3
Bromide SCHEMBL3051472 0.83 STAT3 (0.55) PIK3CAPRKAA2STAT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2207773-B1 HETEROCYCLIC COMPOUND AND PHARMACEUTICAL COMPOSITION THEREOF OTSUKA PHARMA CO LTD (JP) 2012-07-11 EP disclosed
EP-2207773-A2 HETEROCYCLIC COMPOUND AND PHARMACEUTICAL COMPOSITION THEREOF Otsuka Pharmaceutical Co., Ltd. (JP) 2010-07-21 EP disclosed
WO-2009057811-A2 HETEROCYCLIC COMPOUND AND PHARMACEUTICAL COMPOSITION THEREOF OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2009-05-07 WO disclosed