SCHEMBL3709926

SCHEMBL3709926

CC(NC(=O)C(F)(F)F)c1ccccc1Br

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.59
PDK1 Q15118 1/20 0.44
PDK2 Q15119 1/20 0.44
PDK3 Q15120 1/20 0.44
PDK4 Q16654 1/20 0.44
LMNA P02545 1/20 0.42
HDAC3 O15379 3/20 0.40
HDAC1 Q13547 3/20 0.40
HDAC6 Q9UBN7 3/20 0.40
CYP2C9 P11712 2/20 0.40
CYP2C19 P33261 1/20 0.39
ESR1 P03372 1/20 0.39
KCNH2 Q12809 1/20 0.39
ALDH1A1 P00352 3/20 0.38
ANPEP P15144 1/20 0.38
HDAC4 P56524 2/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
CNR1 P21554 2/20 0.37
TDP1 Q9NUW8 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17007872 1.00 HTT (0.59) HTTPDK1PDK2PDK3PDK4
SCHEMBL25403697 0.86 ESR1 (0.45) HTTPDK1PDK2PDK3PDK4
SCHEMBL18361484 0.82 GABRA1 (0.46) HTTLMNAHDAC3HDAC1HDAC6
SCHEMBL23381716 0.81 ESR1 (0.51) HTTHDAC3HDAC1HDAC6CYP2C9
SCHEMBL3780674 0.80 PDK1 (0.45) HTTPDK1PDK2PDK3PDK4
SCHEMBL1345465 0.80 HTT (0.66) HTTLMNACYP2C9CYP2C19ALDH1A1
SCHEMBL28974132 0.80 HTT (0.66) HTTLMNACYP2C9CYP2C19ALDH1A1
SCHEMBL17018471 0.80 HTT (0.66) HTTLMNACYP2C9CYP2C19ALDH1A1
SCHEMBL29150632 0.79 CNR1 (0.43) HTTLMNACYP2C9CYP2C19ALDH1A1
SCHEMBL11529099 0.78 HDAC3 (0.63) LMNAHDAC3HDAC1HDAC6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114901652-A Substituted saturated and unsaturated N-heterocyclic carboxamides and related compounds for the treatment of medical disorders 比亚尔R&D投资股份公司 2022-08-12 CN disclosed
CN-104822680-B Imidazopyridine 安斯泰来制药株式会社 2016-10-12 CN disclosed
CN-104822680-A Imidazopyridine compound ASTELLAS PHARMA INC 2015-08-05 CN disclosed
WO-2010084090-A1 PYRIDYL-AZA(THIO)XANTHONE SENSITIZER COMPRISING LANTHANIDE(III) ION COMPLEXING COMPOUNDS, THEIR LUMINESCENT LANTHANIDE (III) ION COMPLEXES AND USE THEREOF AS FLUORESCENT LABELS. CIS BIO INTERNATIONAL (FR) 2010-07-29 WO disclosed