SCHEMBL3780674

SCHEMBL3780674

CC(NC(=O)C(F)(F)F)c1ccccc1C#N

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 1/20 0.45
PDK2 Q15119 1/20 0.45
PDK3 Q15120 1/20 0.45
PDK4 Q16654 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.41
MAPK1 P28482 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39
HTT P42858 1/20 0.38
HDAC3 O15379 1/20 0.38
CYP2C9 P11712 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
ABCC9 O60706 2/20 0.38
ABCC8 Q09428 2/20 0.38
KCNJ11 Q14654 2/20 0.38
KCNJ8 Q15842 2/20 0.38
ESR1 P03372 1/20 0.36
KCNH2 Q12809 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17007872 0.80 HTT (0.59) PDK1PDK2PDK3PDK4MAPK1
SCHEMBL3709926 0.80 HTT (0.59) PDK1PDK2PDK3PDK4MAPK1
SCHEMBL18361484 0.78 GABRA1 (0.46) ALDH1A1LMNAHTTHDAC3CYP2C9
SCHEMBL23381716 0.77 ESR1 (0.51) ALDH1A1HTTHDAC3CYP2C9HDAC1
SCHEMBL11529099 0.75 HDAC3 (0.63) LMNAHDAC3CYP2C9HDAC1HDAC6
SCHEMBL15760882 0.73 GUCY1B2 (0.40) ALDH1A1HTTHDAC3CYP2C9HDAC1
SCHEMBL17021753 0.73 HDAC3 (0.38) HTTHDAC3CYP2C9HDAC1HDAC6
SCHEMBL15760884 0.73 GUCY1B2 (0.40) ALDH1A1HTTHDAC3CYP2C9HDAC1
SCHEMBL3678697 0.73 L3MBTL1 (0.43) L3MBTL1MAPK1SMN1; SMN2ALDH1A1LMNA
SCHEMBL3678695 0.73 L3MBTL1 (0.43) L3MBTL1MAPK1SMN1; SMN2ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010084090-A1 PYRIDYL-AZA(THIO)XANTHONE SENSITIZER COMPRISING LANTHANIDE(III) ION COMPLEXING COMPOUNDS, THEIR LUMINESCENT LANTHANIDE (III) ION COMPLEXES AND USE THEREOF AS FLUORESCENT LABELS. CIS BIO INTERNATIONAL (FR) 2010-07-29 WO disclosed