SCHEMBL3710698

SCHEMBL3710698

COC(=O)CC(O)(CCN(C(=O)OC)[C@@](C)(I)c1ccc(Cl)cc1)c1ccccc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCL2 P10415 2/20 0.39
HTT P42858 2/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
LMNA P02545 2/20 0.34
ALDH1A1 P00352 2/20 0.34
GRIN2D O15399 1/20 0.34
GRIN3B O60391 1/20 0.34
GRIN1 Q05586 1/20 0.34
GRIN2A Q12879 1/20 0.34
GRIN2B Q13224 1/20 0.34
GRIN2C Q14957 1/20 0.34
GRIN3A Q8TCU5 1/20 0.34
KMT2A Q03164 5/20 0.33
L3MBTL1 Q9Y468 2/20 0.33
TDP1 Q9NUW8 1/20 0.33
KCNN4 O15554 1/20 0.33
OPRM1 P35372 1/20 0.32
OPRL1 P41146 1/20 0.32
MIF P14174 1/20 0.32
MEN1 O00255 3/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3717915 0.89 KMT2A (0.34) SMN1; SMN2ALDH1A1KMT2AL3MBTL1TDP1
SCHEMBL3646232 0.89 BCL2 (0.39) BCL2HTTSMN1; SMN2LMNAALDH1A1
SCHEMBL3646047 0.80 KMT2A (0.43) ALDH1A1GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL1846565 0.79 ALDH1A1 (0.34) ALDH1A1KMT2AL3MBTL1TDP1KCNN4
SCHEMBL958265 0.77 UTS2R (0.39) BCL2KMT2AL3MBTL1MEN1
SCHEMBL1844871 0.71 TAAR1 (0.38) KCNN4
SCHEMBL24451337 0.69 KCNN4 (0.49) HTTSMN1; SMN2LMNAALDH1A1KMT2A
SCHEMBL3645623 0.69 KMT2A (0.43) SMN1; SMN2ALDH1A1KMT2AMEN1CYP1A2
SCHEMBL15949367 0.69 UTS2R (0.39) BCL2
SCHEMBL2546997 0.68 ALDH1A1 (0.40) HTTSMN1; SMN2LMNAALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2393807-A1 CYCLIC INHIBITORS OF 11 -HYDROXYSTEROID DEHYDROGENASE 1 Boehringer Ingelheim International GmbH (DE) 2011-12-14 EP disclosed
WO-2010089303-A1 CYCLIC INHIBITORS OF 11 β-HYDROXYSTEROID DEHYDROGENASE 1 BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-08-12 WO disclosed