SCHEMBL364644

SCHEMBL364644

Cc1ccccc1C(C/C(=N\O)c1c[nH]c(=O)c(C)c1)c1ccc(C(=O)NC2(CO)CC2)cc1

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 6/20 0.45
BRD4 O60885 1/20 0.36
EPHX2 P34913 1/20 0.32
CTSA P10619 4/20 0.31
MAPK8 P45983 1/20 0.31
SMN1; SMN2 Q16637 2/20 0.31
TP53 P04637 1/20 0.31
MGAM O43451 1/20 0.30
GAA P10253 1/20 0.30
SI P14410 1/20 0.30
MGAM2 Q2M2H8 1/20 0.30
SLC6A9 P48067 1/20 0.30
KDM4E B2RXH2 1/20 0.30
MAPT P10636 1/20 0.30
TDP1 Q9NUW8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL362661 0.90 BRD4 (0.38) GPBAR1BRD4EPHX2CTSAMAPK8
SCHEMBL364032 0.84 GPBAR1 (0.47) GPBAR1BRD4EPHX2SMN1; SMN2SLC6A9
SCHEMBL363678 0.84 GPBAR1 (0.61) GPBAR1BRD4CTSAMGAMGAA
SCHEMBL362542 0.84 GPBAR1 (0.47) GPBAR1BRD4CTSASMN1; SMN2SLC6A9
SCHEMBL361767 0.84 GPBAR1 (0.47) GPBAR1BRD4CTSASMN1; SMN2SLC6A9
SCHEMBL362350 0.84 GPBAR1 (0.48) GPBAR1BRD4EPHX2CTSASMN1; SMN2
SCHEMBL362310 0.83 GPBAR1 (0.46) GPBAR1BRD4CTSASMN1; SMN2MGAM
SCHEMBL363734 0.82 GPBAR1 (0.45) GPBAR1BRD4CTSASMN1; SMN2SLC6A9
SCHEMBL363430 0.82 GPBAR1 (0.45) GPBAR1BRD4CTSASMN1; SMN2SLC6A9
SCHEMBL1390107 0.82 GPBAR1 (0.46) GPBAR1BRD4MAPK8SMN1; SMN2TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP claimed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO claimed
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed