SCHEMBL371180

SCHEMBL371180

CCOC(=O)Cc1c(C)[nH]c2c1COCC2

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.37
KDM4E B2RXH2 5/20 0.36
HSD17B10 Q99714 2/20 0.36
ALDH1A1 P00352 1/20 0.36
HPGD P15428 1/20 0.36
AKT1 P31749 1/20 0.36
KMT2A Q03164 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
GAA P10253 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
LMNA P02545 3/20 0.34
CYP2C9 P11712 1/20 0.34
ABCB1 P08183 1/20 0.34
TSHR P16473 2/20 0.33
USP2 O75604 1/20 0.33
HCAR2 Q8TDS4 1/20 0.33
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3343330 0.80 LMNA (0.45) MAPK1KDM4EHSD17B10ALDH1A1HPGD
SCHEMBL3344033 0.79 LMNA (0.47) MAPK1KDM4EHSD17B10ALDH1A1HPGD
SCHEMBL17629578 0.68 LMNA (0.68) KDM4EALDH1A1HPGDKMT2ASMN1; SMN2
SCHEMBL25664507 0.66 GAA (0.57) MAPK1KDM4EHSD17B10ALDH1A1KMT2A
SCHEMBL5951427 0.66 HCAR2 (0.44) KDM4EALDH1A1KMT2AL3MBTL1HCAR2
SCHEMBL12818018 0.64 MGAM (0.44) HSD17B10ALDH1A1AKT1GAASMN1; SMN2
SCHEMBL5398985 0.63 MAPK1 (0.64) MAPK1ALDH1A1HPGDKMT2AGAA
SCHEMBL10268198 0.63 HRH3 (0.42) KDM4EHSD17B10ALDH1A1HPGDKMT2A
SCHEMBL6273007 0.62 ALDH1A1 (0.45) MAPK1KDM4EHSD17B10ALDH1A1HPGD
SCHEMBL1564682 0.62 SMN1; SMN2 (0.38) ALDH1A1AKT1KMT2AGAAL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2516416-A1 CRTH2 MODULATORS Ironwood Pharmaceuticals, Inc. (US) 2012-10-31 EP disclosed
WO-2012009134-A1 CRTH2 MODULATORS IRONWOOD PHARMACEUTICALS, INC. (US) 2012-01-19 WO disclosed
WO-2011079007-A1 CRTH2 MODULATORS IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-30 WO disclosed