SCHEMBL3712349

SCHEMBL3712349

CC1(C)CNCCN1C(=O)c1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.54
MAPK1 P28482 1/20 0.47
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
USP2 O75604 1/20 0.42
ALDH1A1 P00352 1/20 0.42
TSHR P16473 1/20 0.42
HSD17B10 Q99714 1/20 0.42
HPGD P15428 1/20 0.41
ACHE P22303 1/20 0.41
CHRNB2 P17787 2/20 0.40
CHRNB4 P30926 2/20 0.40
CHRNA3 P32297 2/20 0.40
CHRNA7 P36544 2/20 0.40
CHRNA4 P43681 2/20 0.40
BLM P54132 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4249148 0.84 MGLL (0.41) SIGMAR1
SCHEMBL31132514 0.82 TSHR (0.36) SIGMAR1MAPK1MEN1KMT2AALDH1A1
SCHEMBL27678060 0.79 SIGMAR1 (0.51) SIGMAR1MAPK1MEN1KMT2AUSP2
SCHEMBL6012279 0.79 SIGMAR1 (0.55) SIGMAR1USP2ALDH1A1TSHRHSD17B10
SCHEMBL31132746 0.79 KMT2A (0.41) KMT2AALDH1A1HPGD
SCHEMBL27696613 0.78 SIGMAR1 (0.50) SIGMAR1MAPK1MEN1KMT2AUSP2
SCHEMBL27626264 0.76 SIGMAR1 (0.44) SIGMAR1MAPK1MEN1KMT2AUSP2
SCHEMBL4107014 0.76 MAPK1 (0.57) SIGMAR1MAPK1MEN1KMT2AUSP2
SCHEMBL1502938 0.76 SOS1 (0.31)
SCHEMBL15034009 0.76 HPGD (0.36) SIGMAR1USP2ALDH1A1TSHRHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010102663-A1 PIPERAZINE DERIVATIVES FOR USE IN THERAPY GLAXO GROUP LIMITED (GB) 2010-09-16 WO disclosed