SCHEMBL3712362

SCHEMBL3712362

CC(C)n1nnnc1CCNC(=O)O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.46
CYP2C19 P33261 2/20 0.46
MEN1 O00255 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C9 P11712 1/20 0.46
KMT2A Q03164 1/20 0.46
ALDH1A1 P00352 4/20 0.40
TRPV1 Q8NER1 2/20 0.37
GAA P10253 2/20 0.35
NPC1 O15118 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
POLB P06746 2/20 0.35
CASP1 P29466 1/20 0.35
RAB9A P51151 1/20 0.35
USP2 O75604 1/20 0.34
DAGLA Q9Y4D2 3/20 0.34
TP53 P04637 1/20 0.34
HPGD P15428 1/20 0.33
HCAR3 P49019 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1779273 0.69 MAPK1 (0.46) ALDH1A1GAANPC1SMN1; SMN2POLB
SCHEMBL18839655 0.69 ALDH1A1 (0.39) MEN1KMT2AALDH1A1TRPV1GAA
SCHEMBL15017837 0.68 TP53 (0.40) MEN1KMT2ATRPV1SMN1; SMN2RAB9A
SCHEMBL28711299 0.68 ALDH1A1 (0.40) CYP1A2CYP2C19MEN1CYP3A4CYP2D6
SCHEMBL18839929 0.68 NAALAD2 (0.38) MEN1KMT2AALDH1A1TRPV1GAA
SCHEMBL3709122 0.67 MAPK1 (0.37) CYP1A2CYP2C19MEN1CYP2C9KMT2A
SCHEMBL10675456 0.65 L3MBTL1 (0.39) CYP1A2CYP2C19MEN1CYP3A4CYP2D6
SCHEMBL28976472 0.64 HCAR3 (0.42) CYP1A2CYP2C19MEN1CYP3A4CYP2D6
SCHEMBL3869686 0.64 DAGLA (0.38) ALDH1A1DAGLA
SCHEMBL4237037 0.64 HTT (0.39) CYP2C19CYP2D6KMT2AALDH1A1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010100144-A1 FUSED BICYCLIC COMPOUNDS AS INHIBITORS FOR PI3 KINASE MERCK SERONO S.A. (CH) 2010-09-10 WO disclosed