SCHEMBL371298

SCHEMBL371298

COc1ccc(C(CC=O)(c2ccc(Br)cc2)c2ccccc2F)cn1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 1/20 0.35
SLC22A12 Q96S37 1/20 0.34
GPR183 P32249 4/20 0.32
CETP P11597 1/20 0.32
TSHR P16473 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
KCNH2 Q12809 1/20 0.31
GUCY1B2 O75343 1/20 0.31
GUCY1A2 P33402 1/20 0.31
GUCY1A1 Q02108 1/20 0.31
GUCY1B1 Q02153 1/20 0.31
HPGD P15428 1/20 0.31
EPHB4 P54760 1/20 0.31
EDNRB P24530 1/20 0.31
EDNRA P25101 1/20 0.31
TRPM8 Q7Z2W7 1/20 0.31
THRB P10828 1/20 0.31
DGAT1 O75907 1/20 0.31
MEN1 O00255 2/20 0.30
KMT2A Q03164 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL362960 0.86 ERN1 (0.36) ERN1GPR183KCNH2THRB
SCHEMBL362683 0.85 ERN1 (0.38) ERN1GPR183THRBMEN1KMT2A
SCHEMBL365266 0.81 ERN1 (0.35) ERN1SMN1; SMN2MEN1KMT2ANPC1
SCHEMBL363777 0.80 KMT2A (0.39) CETPTSHRSMN1; SMN2KCNH2HPGD
SCHEMBL364766 0.75 GPR183 (0.33) GPR183KCNH2
SCHEMBL363931 0.74 TSHR (0.39) SLC22A12TSHRSMN1; SMN2KCNH2MEN1
SCHEMBL362569 0.66 RORA (0.32)
SCHEMBL362479 0.65 HDAC3 (0.30)
SCHEMBL364417 0.65
SCHEMBL363964 0.65 GPR183 (0.38) SLC22A12GPR183SMN1; SMN2KCNH2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed