SCHEMBL3713155

SCHEMBL3713155

COC(=O)c1cc(Cl)nc(NC2CCOCC2)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.41
LRRK2 Q5S007 1/20 0.41
OPRK1 P41145 1/20 0.40
MAPK1 P28482 4/20 0.40
MAPK3 P27361 2/20 0.40
PIK3CA P42336 1/20 0.39
PIK3CB P42338 1/20 0.39
HDAC3 O15379 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
ALDH1A1 P00352 3/20 0.39
KDM4E B2RXH2 1/20 0.39
HPGDS O60760 1/20 0.38
PDE4B Q07343 1/20 0.38
CCNE1 P24864 4/20 0.37
CDK2 P24941 4/20 0.37
CCNT1 O60563 1/20 0.37
RPS6KA1 Q15418 1/20 0.37
HSD17B10 Q99714 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2419105 0.84 TDP1 (0.41) TDP1ALDH1A1KDM4EHPGDSCCNT1
SCHEMBL21143647 0.82 IDH1 (0.45) TDP1ALDH1A1KDM4EHSD17B10
SCHEMBL2024072 0.81 MAPK1 (0.41) LRRK2OPRK1MAPK1MAPK3CCNE1
SCHEMBL31330409 0.79 LRRK2 (0.51) LRRK2OPRK1MAPK1MAPK3HDAC3
SCHEMBL23304492 0.77 TDP1 (0.44) TDP1LRRK2MAPK1KDM4E
SCHEMBL2414787 0.77 ALDH1A1 (0.52) MAPK1ALDH1A1CDK2CCNT1
SCHEMBL569249 0.74 ALDH1A1 (0.59) TDP1ALDH1A1KDM4E
SCHEMBL3715743 0.74 ALDH1A1 (0.50) TDP1ALDH1A1KDM4E
SCHEMBL23684534 0.73 HCAR3 (0.54) TDP1LRRK2MAPK1KDM4ECDK2
SCHEMBL17113096 0.73 HSD17B10 (0.44) LRRK2OPRK1HDAC3HDAC1HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010100475-A1 HYDROXAMIC ACID DERIVATIVES AS GRAM-NEGATIVE ANTIBACTERIAL AGENTS ASTRAZENECA AB (SE) 2010-09-10 WO disclosed
WO-2010100475-A1 HYDROXAMIC ACID DERIVATIVES AS GRAM-NEGATIVE ANTIBACTERIAL AGENTS ASTRAZENECA AB (SE) 2010-09-10 WO disclosed