SCHEMBL3713341

SCHEMBL3713341

CC1(C)COB(c2ccc(C#Cc3cccnc3)cc2)OC1

nearest known ligand 0.49

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 9/20 0.44
CHRNB2 P17787 3/20 0.40
CHRNA4 P43681 3/20 0.40
CYP2A6 P11509 5/20 0.40
CYP2C9 P11712 2/20 0.40
CYP2B6 P20813 2/20 0.40
CYP2C19 P33261 2/20 0.40
FFAR1 O14842 1/20 0.40
CYP2D6 P10635 2/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2E1 P05181 1/20 0.39
CYP3A4 P08684 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3797332 0.86 GRM5 (0.47) GRM5
SCHEMBL3788618 0.85 SNCA (0.38) GRM5FFAR1
SCHEMBL3788621 0.85 APP (0.40) GRM5
SCHEMBL3790314 0.81 LPL (0.46) GRM5CHRNB2CHRNA4CYP2A6CYP2C9
SCHEMBL4078174 0.79 MAPT (0.36) CHRNB2CHRNA4CYP2A6CYP1A2CYP3A4
SCHEMBL3721364 0.78 FFAR1 (0.40) GRM5FFAR1CYP1A2
SCHEMBL13188238 0.78 CYP2A6 (0.46) CYP2A6CYP2C9CYP2C19CYP2D6CYP1A2
SCHEMBL3786338 0.77 GRM5 (0.37) GRM5CYP1A2
SCHEMBL4264297 0.74 SNCA (0.44)
SCHEMBL13907278 0.74 CYP2A6 (0.62) GRM5CHRNB2CHRNA4CYP2A6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010100475-A1 HYDROXAMIC ACID DERIVATIVES AS GRAM-NEGATIVE ANTIBACTERIAL AGENTS ASTRAZENECA AB (SE) 2010-09-10 WO disclosed