SCHEMBL3713623

SCHEMBL3713623

COC(=O)c1cc(-c2ccc(OCc3ccccc3)cc2)ccn1

nearest known ligand 0.57

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 5/20 0.57
NPC1 O15118 2/20 0.51
RAB9A P51151 2/20 0.51
SMN1; SMN2 Q16637 2/20 0.51
SMPD1 P17405 1/20 0.51
MEN1 O00255 1/20 0.51
KMT2A Q03164 1/20 0.51
MAOB P27338 1/20 0.49
GSTP1 P09211 1/20 0.49
GSK3B P49841 1/20 0.48
ACACB O00763 1/20 0.48
MDM2 Q00987 1/20 0.48
NR4A2 P43354 2/20 0.48
ALDH1A1 P00352 1/20 0.48
LMNA P02545 1/20 0.48
HPGD P15428 1/20 0.48
FFAR1 O14842 1/20 0.48
NR4A1 P22736 1/20 0.48
NR4A3 Q92570 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20510001 0.87 LMNA (0.52) NPC1RAB9ASMN1; SMN2SMPD1MEN1
SCHEMBL13188268 0.85 EGFR (0.51) NR4A2ALDH1A1
SCHEMBL3715274 0.85 SMPD1 (0.67) MCL1SMPD1GSTP1
SCHEMBL3712925 0.84 ACACB (0.58) NPC1RAB9ASMN1; SMN2MEN1KMT2A
SCHEMBL3717976 0.84 MCL1 (0.52) MCL1SMN1; SMN2ACACBALDH1A1HPGD
SCHEMBL29735406 0.83 ALDH1A1 (0.51) NR4A2ALDH1A1LMNAHPGD
SCHEMBL3712306 0.83 ALDH1A1 (0.51) NR4A2ALDH1A1LMNAHPGD
SCHEMBL3713517 0.82 NPC1 (0.54) NPC1RAB9ASMN1; SMN2ALDH1A1HPGD
SCHEMBL31580478 0.81 NR1H4 (0.61) NPC1RAB9ASMN1; SMN2MEN1KMT2A
SCHEMBL9343582 0.81 SMN1; SMN2 (0.65) NPC1RAB9ASMN1; SMN2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010100475-A1 HYDROXAMIC ACID DERIVATIVES AS GRAM-NEGATIVE ANTIBACTERIAL AGENTS ASTRAZENECA AB (SE) 2010-09-10 WO disclosed
WO-2010100475-A1 HYDROXAMIC ACID DERIVATIVES AS GRAM-NEGATIVE ANTIBACTERIAL AGENTS ASTRAZENECA AB (SE) 2010-09-10 WO disclosed