SCHEMBL3713658

SCHEMBL3713658

COC(=O)c1cc(-c2ccc(C#Cc3cccnc3)cc2)cnc1N1CC(O)C1

nearest known ligand 0.40

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
OPRK1 P41145 17/20 0.40
AAK1 Q2M2I8 1/20 0.38
NR4A2 P43354 1/20 0.38
ABL1 P00519 1/20 0.38
OPRM1 P35372 1/20 0.37
OPRD1 P41143 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13188575 0.88 NR4A2 (0.48) OPRK1NR4A2ABL1
SCHEMBL3711625 0.88 FFAR1 (0.36) AAK1ABL1
SCHEMBL3715549 0.87 OPRK1 (0.44) OPRK1AAK1NR4A2
SCHEMBL3715130 0.87 OPRK1 (0.45) OPRK1ABL1OPRM1OPRD1
SCHEMBL3711387 0.81 AAK1 (0.45) AAK1NR4A2
SCHEMBL3717587 0.80 AAK1 (0.42) AAK1NR4A2
SCHEMBL3713123 0.80 IKBKE (0.51) AAK1NR4A2ABL1
SCHEMBL3715859 0.79 AAK1 (0.44) AAK1NR4A2
SCHEMBL3709369 0.78 AAK1 (0.41) AAK1NR4A2
SCHEMBL3714045 0.77 CYP19A1 (0.41) AAK1ABL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010100475-A1 HYDROXAMIC ACID DERIVATIVES AS GRAM-NEGATIVE ANTIBACTERIAL AGENTS ASTRAZENECA AB (SE) 2010-09-10 WO disclosed