SCHEMBL3713722

SCHEMBL3713722

CCc1ccc2cccc(OC3CCN(C(=O)OC(C)(C)C)CC3)c2n1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 1/20 0.50
GPR119 Q8TDV5 10/20 0.49
PDE4D Q08499 3/20 0.48
PDE4A P27815 2/20 0.48
PDE4B Q07343 2/20 0.48
PDE4C Q08493 2/20 0.48
CACNB4 O00305 2/20 0.45
CACNA1A O00555 2/20 0.45
CACNA1G O43497 2/20 0.45
CACNG3 O60359 2/20 0.45
CACNA1F O60840 2/20 0.45
CACNA1H O95180 2/20 0.45
CACNB3 P54284 2/20 0.45
CACNA2D1 P54289 2/20 0.45
CACNG7 P62955 2/20 0.45
CACNA1B Q00975 2/20 0.45
CACNA1D Q01668 2/20 0.45
CACNB1 Q02641 2/20 0.45
CACNG1 Q06432 2/20 0.45
CACNB2 Q08289 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3706690 0.86 KDM1A (0.52) KDM1AGPR119PDE4DPDE4APDE4B
SCHEMBL3718944 0.84 GPR119 (0.42) GPR119PIM1PIM2
SCHEMBL3805418 0.83 KDM1A (0.53) KDM1AGPR119PDE4DPDE4APDE4B
SCHEMBL1632232 0.80 KDM1A (0.50) KDM1AGPR119PDE4DPDE4APDE4B
SCHEMBL5454387 0.78 GPR119 (0.57) KDM1AGPR119PDE4DPDE4APDE4B
SCHEMBL3714938 0.78 KDM1A (0.50) KDM1AGPR119PDE4DPDE4APDE4B
SCHEMBL213729 0.76 KDM1A (0.56) KDM1AGPR119PDE4DPDE4APDE4B
SCHEMBL1975955 0.76 PIM2 (0.77) PIM1PIM2
Hydrochloric Acid SCHEMBL215238 0.76 KDM1A (0.55) KDM1AGPR119PDE4DPDE4APDE4B
SCHEMBL3711289 0.75 HRH1 (0.52) PDE4DPDE4APDE4BPDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010094643-A1 QUINOLINE DERIVATIVES AND THEIR USES FOR RHINITIS AND URTICARIA GLAXO GROUP LIMITED (GB) 2010-08-26 WO disclosed