SCHEMBL3714938

SCHEMBL3714938

Cc1cnc2c(OC3CCN(C(=O)OC(C)(C)C)CC3)cccc2c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 1/20 0.50
NPBWR1 P48145 1/20 0.48
MCHR1 Q99705 1/20 0.48
GPR119 Q8TDV5 9/20 0.47
PDE4B Q07343 3/20 0.46
PDE4A P27815 2/20 0.46
PDE4C Q08493 2/20 0.46
PDE4D Q08499 2/20 0.46
PIK3CD O00329 2/20 0.45
CACNB4 O00305 1/20 0.44
CACNA1A O00555 1/20 0.44
CACNA1G O43497 1/20 0.44
CACNG3 O60359 1/20 0.44
CACNA1F O60840 1/20 0.44
CACNA1H O95180 1/20 0.44
CACNB3 P54284 1/20 0.44
CACNA2D1 P54289 1/20 0.44
CACNG7 P62955 1/20 0.44
CACNA1B Q00975 1/20 0.44
CACNA1D Q01668 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3709887 0.86 GPR119 (0.48) KDM1ANPBWR1MCHR1GPR119PDE4B
SCHEMBL3805418 0.85 KDM1A (0.53) KDM1AGPR119PDE4BPDE4APDE4C
SCHEMBL3714939 0.83 GPR119 (0.46) GPR119PDE4BPIK3CD
SCHEMBL3706690 0.82 KDM1A (0.52) KDM1AGPR119PDE4BPDE4APDE4C
SCHEMBL1632232 0.82 KDM1A (0.50) KDM1ANPBWR1MCHR1GPR119PDE4B
SCHEMBL3708948 0.80 GPR119 (0.51) KDM1AGPR119PDE4BPDE4APDE4C
SCHEMBL3055131 0.79 GPR119 (0.47) KDM1AGPR119PDE4BPDE4APDE4C
SCHEMBL1149124 0.79 CACNB4 (0.49) KDM1ANPBWR1MCHR1GPR119PDE4B
SCHEMBL5665583 0.78 KDM1A (0.51) KDM1ANPBWR1MCHR1GPR119PDE4B
SCHEMBL3717757 0.78 KDM1A (0.51) KDM1AGPR119PDE4BPDE4APDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010094643-A1 QUINOLINE DERIVATIVES AND THEIR USES FOR RHINITIS AND URTICARIA GLAXO GROUP LIMITED (GB) 2010-08-26 WO disclosed