SCHEMBL3713792

SCHEMBL3713792

[CH2]c1cccc(-c2ccccc2F)c1-c1cccc2ccccc12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHFR P00374 1/20 0.41
AKR1C3 P42330 1/20 0.38
AKR1C2 P52895 1/20 0.38
TYMP P19971 1/20 0.36
CYP1A1 P04798 3/20 0.36
CYP1A2 P05177 3/20 0.36
CYP1B1 Q16678 3/20 0.36
AHR P35869 2/20 0.36
PRKDC P78527 1/20 0.36
DNMT1 P26358 1/20 0.36
MAPT P10636 1/20 0.36
NPC1 O15118 2/20 0.35
MEN1 O00255 1/20 0.35
RAB9A P51151 1/20 0.35
KMT2A Q03164 1/20 0.35
ADORA2A P29274 1/20 0.35
HPRT1 P00492 1/20 0.34
KDM4E B2RXH2 1/20 0.33
PTPN1 P18031 1/20 0.33
CES1 P23141 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2491515 0.87 DHFR (0.46) DHFRTYMPCYP1A2DNMT1KDM4E
SCHEMBL2495765 0.85 HTR1A (0.35) MAPTNPC1MEN1RAB9AKMT2A
SCHEMBL3153748 0.81 AKR1C3 (0.49) AKR1C3AKR1C2CYP1A1CYP1A2CYP1B1
SCHEMBL30002959 0.81 AKR1C3 (0.49) AKR1C3AKR1C2CYP1A1CYP1A2CYP1B1
SCHEMBL2030385 0.80 CYP17A1 (0.43) DHFRTYMPCYP1A2ADORA2AKDM4E
SCHEMBL22978397 0.80 NPC1 (0.43) DHFRAKR1C3AKR1C2TYMPCYP1A1
SCHEMBL28779511 0.79 AKR1C3 (0.40) DHFRAKR1C3AKR1C2TYMPCYP1A1
SCHEMBL28232750 0.79 DHFR (0.44) DHFRAKR1C3AKR1C2TYMPCYP1A1
SCHEMBL29104508 0.79 AKR1C3 (0.47) AKR1C3AKR1C2CYP1A1CYP1A2CYP1B1
SCHEMBL29165700 0.73 DHFR (0.39) DHFRAKR1C3AKR1C2CYP1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2398815-A2 SYNTHESIS OF ARA-2'-O-METHYL-NUCLEOSIDES, CORRESPONDING PHOSPHORAMIDITES AND OLIGONUCLEOTIDES INCORPORATING NOVEL MODIFICATIONS FOR BIOLOGICAL APPLICATION IN THERAPEUTICS, DIAGNOSTICS, G- TETRAD FORMING OLIGONUCLEOTIDES AND APTAMERS Chemgenes Corporation (US) 2011-12-28 EP disclosed
WO-2010096201-A2 SYNTHESIS OF ARA-2'-O-METHYL-NUCLEOSIDES, CORRESPONDING PHOSPHORAMIDITES AND OLIGONUCLEOTIDES INCORPORATING NOVEL MODIFICATIONS FOR BIOLOGICAL APPLICATION IN THERAPEUTICS, DIAGNOSTICS, G- TETRAD FORMING OLIGONUCLEOTIDES AND APTAMERS CHEMGENES CORPORATION (US) 2010-08-26 WO disclosed