SCHEMBL3715260

SCHEMBL3715260

Cc1csc(C(=O)O)c1NC(=O)C(F)(F)F

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.52
KMT2A Q03164 1/20 0.52
L3MBTL1 Q9Y468 3/20 0.45
MAPT P10636 1/20 0.43
PKM P14618 1/20 0.43
ATM Q13315 1/20 0.43
POLB P06746 2/20 0.41
TDP1 Q9NUW8 1/20 0.41
CYP1A2 P05177 2/20 0.41
CYP3A4 P08684 2/20 0.41
CYP2C19 P33261 1/20 0.41
HTR1A P08908 1/20 0.37
SCN1A P35498 1/20 0.37
SCN2A Q99250 1/20 0.37
SCN3A Q9NY46 1/20 0.37
GPR35 Q9HC97 1/20 0.36
PDK1 Q15118 1/20 0.35
PDK2 Q15119 1/20 0.35
PDK3 Q15120 1/20 0.35
PDK4 Q16654 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL613613 0.84 MAPT (0.58) ALDH1A1KMT2AMAPTPKMATM
SCHEMBL21813827 0.79 CYP1A2 (0.45) ALDH1A1KMT2AL3MBTL1MAPTPKM
SCHEMBL5234643 0.79 PDK1 (0.42) ALDH1A1KMT2AL3MBTL1MAPTPKM
SCHEMBL6317855 0.78 ALDH1A1 (0.56) ALDH1A1KMT2AL3MBTL1MAPTPKM
SCHEMBL4785611 0.75 ALDH1A1 (0.53) ALDH1A1KMT2AL3MBTL1MAPTPKM
SCHEMBL9098700 0.75 ALDH1A1 (0.53) ALDH1A1KMT2AL3MBTL1MAPTPKM
SCHEMBL23295963 0.74 ALDH1A1 (0.52) ALDH1A1KMT2AL3MBTL1MAPTPKM
SCHEMBL15399918 0.73 PDK1 (0.40) KMT2AL3MBTL1MAPTPOLBCYP1A2
SCHEMBL25095439 0.72 PDK1 (0.55) ALDH1A1KMT2AL3MBTL1MAPTPKM
SCHEMBL7902025 0.72 ALDH1A1 (0.71) ALDH1A1KMT2AL3MBTL1MAPTATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010101302-A1 THIENOPYRIMIDINE AS CDC7 KINASE INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-09-10 WO disclosed