SCHEMBL3716019

SCHEMBL3716019

CCc1ccc2c(c1)C(C)(C)CCN2C(=O)C(F)(F)F

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 2/20 0.42
HDAC6 Q9UBN7 2/20 0.42
RARB P10826 5/20 0.39
RARA P10276 4/20 0.39
RXRA P19793 2/20 0.39
RXRB P28702 1/20 0.39
RXRG P48443 1/20 0.39
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA7 P43166 1/20 0.38
CA9 Q16790 1/20 0.38
RARG P13631 2/20 0.38
CYP26A1 O43174 1/20 0.37
CYP26B1 Q9NR63 1/20 0.37
RORC P51449 2/20 0.36
PDK2 Q15119 1/20 0.36
NR1I2 O75469 1/20 0.36
NR1H2 P55055 1/20 0.36
NR1H3 Q13133 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3788762 0.84 CA12 (0.40) HDAC1HDAC6RARBRARACA12
SCHEMBL3716822 0.79 RXRA (0.38) HDAC1HDAC6RARBRARARXRA
SCHEMBL4430316 0.75 CA12 (0.39) HDAC1HDAC6RARBRARACA12
SCHEMBL6223920 0.75 CA12 (0.36) HDAC1HDAC6RARBRARACA12
SCHEMBL7878918 0.74 CA12 (0.36) HDAC1HDAC6RARBRARARXRA
SCHEMBL4425583 0.73 FFAR4 (0.38) RXRARXRBRXRGCA12CA1
SCHEMBL3799829 0.73 RARA (0.36) HDAC1HDAC6RARBRARARXRA
SCHEMBL11924574 0.72 KDM1A (0.46) HDAC1HDAC6RARBRARARXRA
SCHEMBL13185172 0.70 POLB (0.45) ALDH1A1MAPTHTT
SCHEMBL3717297 0.70 RORC (0.38) HDAC1HDAC6RXRARXRBRXRG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010129467-A1 COMPOUNDS AND METHODS FOR INHIBITION OF RENIN, AND INDICATIONS THEREFOR PLEXXIKON, INC. (US) 2010-11-11 WO disclosed
WO-2010129467-A1 COMPOUNDS AND METHODS FOR INHIBITION OF RENIN, AND INDICATIONS THEREFOR PLEXXIKON, INC. (US) 2010-11-11 WO disclosed