SCHEMBL3716306

SCHEMBL3716306

Nc1ccc(-c2cn[nH]c2)cc1Oc1ccccc1

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 6/20 0.53
AKT2 P31751 2/20 0.50
AKT1 P31749 1/20 0.50
BTK Q06187 1/20 0.44
TNK2 Q07912 1/20 0.43
ALK Q9UM73 1/20 0.42
ROCK1 Q13464 3/20 0.42
CHEK1 O14757 1/20 0.41
MELK Q14680 1/20 0.41
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
GRK2 P25098 1/20 0.39
GRK1 Q15835 1/20 0.39
IKBKB O14920 1/20 0.39
BRAF P15056 1/20 0.39
FEN1 P39748 1/20 0.39
XDH P47989 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30697305 0.84 ALDH1A1 (0.52) CYP1A2CYP3A4CYP2C9CYP2C19IKBKB
SCHEMBL5014782 0.84 ALDH1A1 (0.52) CYP1A2CYP3A4CYP2C9CYP2C19IKBKB
SCHEMBL30393911 0.82 ALDH1A1 (0.50) CYP1A2CYP3A4CYP2C9CYP2C19IKBKB
SCHEMBL3782732 0.81 CYP3A4 (0.49) CYP1A2CYP3A4CYP2C9CYP2C19IKBKB
SCHEMBL3716304 0.80 CTNNB1 (0.52) ROCK2AKT2AKT1ROCK1MELK
SCHEMBL18783247 0.79 AKT2 (0.50) ROCK2AKT2AKT1BTKTNK2
SCHEMBL30394034 0.79 CYP3A4 (0.47) CYP1A2CYP3A4CYP2C9CYP2C19IKBKB
SCHEMBL3722814 0.79 ROCK2 (0.60) ROCK2AKT2AKT1ROCK1MELK
SCHEMBL3656438 0.78 ALDH1A1 (0.67) ROCK2ROCK1CHEK1MELKCYP3A4
SCHEMBL3793152 0.78 MAOA (0.53) CYP1A2CYP3A4CYP2C9CYP2C19IKBKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2234618-A1 BENZOPYRANS AND ANALOGS AS RHO KINASE INHIBITORS The Scripps Research Institute (US) 2010-10-06 EP disclosed
WO-2009079008-A1 BENZOPYRANS AND ANALOGS AS RHO KINASE INHIBITORS FENG YANGBO (US) 2009-06-25 WO disclosed