SCHEMBL3716451

SCHEMBL3716451

O=C(O)[C@@H]1C[C@@H](C(=O)C(c2ccc(Cl)cc2)(N2CCOCC2)S(=O)(=O)c2ccccc2Cl)CN1

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CTSS P25774 6/20 0.36
FAAH O00519 2/20 0.35
KMT2A Q03164 3/20 0.34
CNR1 P21554 1/20 0.34
ALDH1A1 P00352 3/20 0.33
KDM4E B2RXH2 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
EPHX2 P34913 1/20 0.33
MEN1 O00255 1/20 0.32
MAPT P10636 1/20 0.32
HTT P42858 1/20 0.32
DPP4 P27487 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
CTSL P07711 1/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3718248 0.80 HSD11B1 (0.38) FAAHKMT2AALDH1A1EPHX2L3MBTL1
SCHEMBL3718796 0.75 CYP1A2 (0.42) CTSSFAAHALDH1A1DPP4L3MBTL1
SCHEMBL3718974 0.74 KMT2A (0.35) FAAHKMT2AEPHX2
SCHEMBL695114 0.73 CTSS (0.40) CTSSCTSL
SCHEMBL3716343 0.69 CYP1A2 (0.39) DPP4
SCHEMBL3721567 0.69 CYP1A2 (0.39) CTSSFAAHHTTDPP4
SCHEMBL3715962 0.68 SLC1A3 (0.46) CTSSFAAHALDH1A1DPP4L3MBTL1
SCHEMBL4740683 0.66 CTSS (0.55) CTSSKMT2AALDH1A1SMN1; SMN2HTT
SCHEMBL694969 0.66 CTSS (0.43) CTSSFAAHALDH1A1L3MBTL1CTSL
SCHEMBL15327130 0.66 CTSS (0.43) CTSSFAAHALDH1A1L3MBTL1CTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010121918-A1 PROLINE DERIVATIVES AS CATHEPSIN INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2010-10-28 WO disclosed