SCHEMBL3718974

SCHEMBL3718974

CC(CS(=O)(=O)c1ccccc1Cl)(C(=O)[C@H]1CN[C@H](C(=O)O)C1)c1ccc(Cl)cc1

nearest known ligand 0.35

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.35
FNTA P49354 1/20 0.35
PGGT1B P53609 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
ALOX15 P16050 1/20 0.35
CYP2C19 P33261 1/20 0.35
SLC1A3 P43003 1/20 0.35
SLC1A2 P43004 1/20 0.35
SLC1A1 P43005 1/20 0.35
HSD11B1 P28845 12/20 0.33
FAAH O00519 1/20 0.32
ELOVL6 Q9H5J4 1/20 0.32
EPHX2 P34913 1/20 0.32
DRD2 P14416 1/20 0.32
OPRM1 P35372 1/20 0.32
DRD3 P35462 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3721567 0.85 CYP1A2 (0.39) FNTAPGGT1BCYP1A2CYP2D6ALOX15
SCHEMBL3718248 0.81 HSD11B1 (0.38) KMT2AFNTAPGGT1BCYP1A2CYP2D6
SCHEMBL3723534 0.78 CYP2D6 (0.37) CYP1A2CYP2D6ALOX15CYP2C19SLC1A3
SCHEMBL3718796 0.77 CYP1A2 (0.42) CYP1A2CYP2D6ALOX15CYP2C19SLC1A3
SCHEMBL3716451 0.74 CTSS (0.36) KMT2AFAAHEPHX2
SCHEMBL3718799 0.72 ARG1 (0.43) CYP1A2CYP2D6ALOX15CYP2C19SLC1A3
SCHEMBL3715962 0.72 SLC1A3 (0.46) CYP1A2CYP2D6ALOX15CYP2C19SLC1A3
SCHEMBL3716552 0.71 ARG1 (0.47) KMT2ACYP1A2CYP2D6ALOX15CYP2C19
SCHEMBL3716343 0.70 CYP1A2 (0.39) CYP1A2CYP2D6ALOX15CYP2C19SLC1A3
SCHEMBL693779 0.70 CTSL (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010121918-A1 PROLINE DERIVATIVES AS CATHEPSIN INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2010-10-28 WO disclosed