SCHEMBL3716625

SCHEMBL3716625

COCCOc1nc(C(=O)NOC2CCOCC2)cc(-c2ccc(C#Cc3ccc(CN4CCOCC4)cc3)cc2)n1

nearest known ligand 0.44

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TLR7 Q9NYK1 2/20 0.41
ITK Q08881 1/20 0.40
MMP2 P08253 2/20 0.40
MMP8 P22894 2/20 0.40
MMP13 P45452 2/20 0.40
KMT2A Q03164 1/20 0.40
SYK P43405 1/20 0.39
ACVR1 Q04771 1/20 0.38
MMP9 P14780 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13187751 0.91 MAPK14 (0.42) SYK
SCHEMBL3713800 0.88 HDAC1 (0.44) TLR7ITKMMP2MMP8MMP13
SCHEMBL3715177 0.86 TLR7 (0.44) TLR7ITKKMT2A
SCHEMBL3716614 0.81 HDAC1 (0.49) MMP2MMP8MMP13
SCHEMBL3710611 0.81 ACACB (0.47) ITKSYK
SCHEMBL13188373 0.79 HDAC1 (0.46)
SCHEMBL3709560 0.78 KMO (0.50)
SCHEMBL3713318 0.77 KMT2A (0.46) ITKKMT2A
SCHEMBL13188620 0.76 KMO (0.47)
SCHEMBL3713497 0.76 KDM4E (0.40) ITKMMP2MMP8MMP13KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010100475-A1 HYDROXAMIC ACID DERIVATIVES AS GRAM-NEGATIVE ANTIBACTERIAL AGENTS ASTRAZENECA AB (SE) 2010-09-10 WO disclosed