SCHEMBL3717092

SCHEMBL3717092

O=C(O)c1cccc(NS(=O)(=O)c2cc(F)cc(F)c2)c1

nearest known ligand 0.69

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
POLB P06746 4/20 0.69
THRB P10828 1/20 0.65
PFKFB3 Q16875 1/20 0.64
MEN1 O00255 4/20 0.60
KMT2A Q03164 4/20 0.60
MAPT P10636 2/20 0.60
ALDH1A1 P00352 1/20 0.60
LMNA P02545 1/20 0.58
AKR1C3 P42330 1/20 0.56
HSD17B10 Q99714 1/20 0.53
PTK2B Q14289 1/20 0.52
ITGA1 P56199 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3724198 0.90 THRB (0.79) POLBTHRBPFKFB3MEN1KMT2A
SCHEMBL894613 0.84 POLB (0.82) POLBTHRBPFKFB3MEN1KMT2A
SCHEMBL400223 0.84 THRB (0.83) POLBTHRBPFKFB3MEN1KMT2A
SCHEMBL788070 0.81 PFKFB3 (0.83) POLBTHRBPFKFB3MEN1KMT2A
SCHEMBL11025715 0.79 POLB (0.78) POLBTHRBPFKFB3MEN1KMT2A
SCHEMBL17331335 0.79 POLB (0.78) POLBPFKFB3MEN1KMT2AMAPT
SCHEMBL2888070 0.79 POLB (0.94) POLBPFKFB3MEN1KMT2AMAPT
SCHEMBL2241495 0.79 ITGA1 (0.80) POLBPFKFB3MEN1KMT2AMAPT
SCHEMBL30209693 0.79 POLB (0.94) POLBPFKFB3MEN1KMT2AMAPT
SCHEMBL3556551 0.79 THRB (0.65) POLBTHRBPFKFB3MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010126922-A1 BENZIMIDAZOLECARBOXAMIDES AS INHIBITORS OF FAK GLAXOSMITHKLINE LLC (US) 2010-11-04 WO disclosed
WO-2010126922-A1 BENZIMIDAZOLECARBOXAMIDES AS INHIBITORS OF FAK GLAXOSMITHKLINE LLC (US) 2010-11-04 WO disclosed