SCHEMBL3717239

SCHEMBL3717239

c1cnc2c(OC3CCNC3)cccc2c1

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 6/20 0.53
SLC6A2 P23975 6/20 0.53
PIM1 P11309 4/20 0.53
PIM2 Q9P1W9 4/20 0.53
DDB1 Q16531 1/20 0.51
CRBN Q96SW2 1/20 0.51
CHRNB2 P17787 1/20 0.50
CHRNA4 P43681 1/20 0.50
KDM4E B2RXH2 1/20 0.43
PRKCZ Q05513 1/20 0.43
HTR2C P28335 2/20 0.43
HTR2B P41595 2/20 0.43
JAK2 O60674 1/20 0.42
JAK1 P23458 1/20 0.42
TYK2 P29597 1/20 0.42
JAK3 P52333 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1115666 1.00 HTR1A (0.53) HTR1ASLC6A2PIM1PIM2DDB1
SCHEMBL3718465 1.00 HTR1A (0.53) HTR1ASLC6A2PIM1PIM2DDB1
SCHEMBL3715640 0.91 DDB1 (0.53) HTR1ASLC6A2PIM1PIM2DDB1
SCHEMBL21227882 0.88 DDB1 (0.52) HTR1ASLC6A2DDB1CRBNKDM4E
Hydrochloric Acid SCHEMBL21222507 0.87 DDB1 (0.51) HTR1ASLC6A2DDB1CRBNKDM4E
SCHEMBL29506919 0.83 DDB1 (0.56) DDB1CRBNKDM4E
SCHEMBL13137148 0.83 CHRNB2 (0.45) HTR1ASLC6A2PIM1PIM2CHRNB2
SCHEMBL3229084 0.81 PIM1 (0.55) PIM1PIM2DDB1CRBN
SCHEMBL3232275 0.81 PIM1 (0.55) PIM1PIM2DDB1CRBN
SCHEMBL3232268 0.81 PIM1 (0.55) PIM1PIM2DDB1CRBN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010094643-A1 QUINOLINE DERIVATIVES AND THEIR USES FOR RHINITIS AND URTICARIA GLAXO GROUP LIMITED (GB) 2010-08-26 WO disclosed