SCHEMBL3718486

SCHEMBL3718486

CC(C)Oc1ccc(Oc2ccc3cc(CCN)ccc3n2)c(Br)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
NFKB1 P19838 1/20 0.37
KDM4E B2RXH2 1/20 0.36
ATM Q13315 1/20 0.36
LMNA P02545 2/20 0.36
MEN1 O00255 1/20 0.36
APEX1 P27695 1/20 0.36
KMT2A Q03164 1/20 0.36
S1PR3 Q99500 1/20 0.35
S1PR5 Q9H228 1/20 0.35
FFAR4 Q5NUL3 1/20 0.34
TAAR1 Q96RJ0 4/20 0.33
GLA P06280 2/20 0.33
TAAR5 O14804 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
MAPK1 P28482 1/20 0.33
NCF1 P14598 1/20 0.33
TEC P42680 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3718570 0.93 TSHR (0.38) TSHRCYP1A2CYP3A4NFKB1KDM4E
SCHEMBL3720128 0.89 KDM4E (0.45) TSHRCYP1A2CYP3A4NFKB1KDM4E
SCHEMBL3720741 0.88 FFAR4 (0.36) TSHRCYP1A2CYP3A4NFKB1KDM4E
SCHEMBL3720774 0.87 GLA (0.43) TSHRCYP1A2CYP3A4NFKB1KDM4E
SCHEMBL3719835 0.86 FFAR4 (0.36) TSHRCYP1A2CYP3A4NFKB1KDM4E
SCHEMBL3717501 0.86 GLA (0.39) TSHRCYP1A2CYP3A4NFKB1KDM4E
SCHEMBL3717202 0.85 ACACB (0.38) TSHRCYP1A2CYP3A4NFKB1LMNA
SCHEMBL3719552 0.85 PDE3B (0.34) LMNAMEN1KMT2AS1PR3S1PR5
SCHEMBL3719380 0.85 RXRA (0.37) TSHRCYP1A2CYP3A4NFKB1S1PR3
SCHEMBL3722047 0.84 GLA (0.42) TSHRCYP1A2CYP3A4NFKB1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010127208-A1 INHIBITORS OF ACETYL-COA CARBOXYLASE FOREST LABORATORIES HOLDINGS LIMITED (BM) 2010-11-04 WO disclosed