SCHEMBL3717501

SCHEMBL3717501

CCOc1ccc(Oc2ccc3cc(CCN)ccc3n2)c(Br)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GLA P06280 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
CYP3A4 P08684 2/20 0.38
TSHR P16473 2/20 0.38
CYP1A2 P05177 1/20 0.38
NFKB1 P19838 1/20 0.38
KDM4E B2RXH2 3/20 0.37
ATM Q13315 2/20 0.37
LMNA P02545 5/20 0.37
KMT2A Q03164 5/20 0.37
MEN1 O00255 4/20 0.37
APEX1 P27695 1/20 0.37
NCF1 P14598 1/20 0.36
MAPT P10636 3/20 0.35
NPSR1 Q6W5P4 2/20 0.35
HTR2A P28223 1/20 0.35
HTR2C P28335 1/20 0.35
HTR2B P41595 1/20 0.35
ALDH1A1 P00352 1/20 0.35
TP53 P04637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3722047 0.92 GLA (0.42) GLASMN1; SMN2CYP3A4TSHRCYP1A2
SCHEMBL3726083 0.91 GLA (0.39) GLASMN1; SMN2CYP3A4TSHRCYP1A2
SCHEMBL3720106 0.87 SMN1; SMN2 (0.49) GLASMN1; SMN2CYP3A4TSHRCYP1A2
SCHEMBL3718486 0.86 TSHR (0.37) GLASMN1; SMN2CYP3A4TSHRCYP1A2
SCHEMBL3721858 0.86 GLA (0.43) GLASMN1; SMN2CYP3A4TSHRCYP1A2
SCHEMBL3721410 0.85 MAPT (0.36) SMN1; SMN2KDM4EATMLMNAKMT2A
SCHEMBL3719459 0.83 PARP10 (0.37)
SCHEMBL3722996 0.83 MTNR1A (0.53) SMN1; SMN2LMNAMAPTALDH1A1
SCHEMBL3718570 0.83 TSHR (0.38) GLASMN1; SMN2CYP3A4TSHRCYP1A2
SCHEMBL3719435 0.82 TLR8 (0.37) GLASMN1; SMN2CYP3A4TSHRCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010127208-A1 INHIBITORS OF ACETYL-COA CARBOXYLASE FOREST LABORATORIES HOLDINGS LIMITED (BM) 2010-11-04 WO disclosed