SCHEMBL3718906

SCHEMBL3718906

O=C(O)[C@@H]1C[C@@H](C(C(F)(F)C(F)(F)F)S(=O)(=O)c2ccccc2Cl)CN1

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 10/20 0.36
CTSS P25774 1/20 0.35
ABCC9 O60706 1/20 0.34
ABCC8 Q09428 1/20 0.34
KCNJ11 Q14654 1/20 0.34
KCNJ8 Q15842 1/20 0.34
ELOVL6 Q9H5J4 1/20 0.34
GRIK1 P39086 3/20 0.33
GRIA2 P42262 3/20 0.33
CYP1A2 P05177 1/20 0.32
CYP2D6 P10635 1/20 0.32
ALOX15 P16050 1/20 0.32
CYP2C19 P33261 1/20 0.32
SLC1A3 P43003 1/20 0.32
SLC1A2 P43004 1/20 0.32
SLC1A1 P43005 1/20 0.32
FAAH O00519 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3723335 0.91 ELOVL6 (0.35) HSD11B1CTSSELOVL6GRIK1GRIA2
SCHEMBL15327131 0.72 CTSS (0.43) CTSSELOVL6CYP1A2CYP2D6ALOX15
SCHEMBL15327130 0.72 CTSS (0.43) CTSSELOVL6CYP1A2CYP2D6ALOX15
SCHEMBL694969 0.72 CTSS (0.43) CTSSELOVL6CYP1A2CYP2D6ALOX15
SCHEMBL3719416 0.71 ARG1 (0.39) HSD11B1CTSSELOVL6GRIK1CYP1A2
SCHEMBL3715962 0.70 SLC1A3 (0.46) CTSSGRIK1GRIA2CYP1A2CYP2D6
SCHEMBL3718796 0.69 CYP1A2 (0.42) HSD11B1CTSSGRIK1GRIA2CYP1A2
SCHEMBL3717159 0.69 ELOVL6 (0.33) HSD11B1CTSSELOVL6CYP1A2CYP2D6
SCHEMBL3718799 0.69 ARG1 (0.43) CTSSGRIK1CYP1A2CYP2D6ALOX15
SCHEMBL3718924 0.68 SLC6A2 (0.36) GRIK1GRIA2CYP1A2CYP2D6ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010121918-A1 PROLINE DERIVATIVES AS CATHEPSIN INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2010-10-28 WO disclosed