SCHEMBL3719008

SCHEMBL3719008

COc1ccc(Oc2ccc(CNC(=O)C3(N)CC3)nc2)c(C(F)(F)F)c1

nearest known ligand 0.43

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 1/20 0.43
EPHX2 P34913 10/20 0.41
ADORA2A P29274 1/20 0.38
KMT2A Q03164 1/20 0.38
MAPK10 P53779 3/20 0.37
MAPK8 P45983 2/20 0.37
ESRRA P11474 1/20 0.37
AKT2 P31751 1/20 0.37
PTPN7 P35236 1/20 0.37
DUSP3 P51452 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL3725905 0.96 P2RX7 (0.41) P2RX7EPHX2ADORA2AKMT2AMAPK10
SCHEMBL3722862 0.90 P2RX7 (0.43) P2RX7EPHX2MAPK10MAPK8ESRRA
SCHEMBL2549180 0.87 L3MBTL1 (0.45) P2RX7EPHX2PTPN7DUSP3
SCHEMBL13191685 0.87 P2RX7 (0.39) P2RX7EPHX2ADORA2AKMT2AMAPK10
SCHEMBL13191703 0.85 P2RX7 (0.38) P2RX7EPHX2ADORA2AKMT2A
SCHEMBL13191622 0.85 EPHX2 (0.47) P2RX7EPHX2KMT2A
SCHEMBL13191240 0.84 EPHX2 (0.43) P2RX7EPHX2KMT2A
SCHEMBL13191684 0.84 EPHX2 (0.39) P2RX7EPHX2
SCHEMBL13191618 0.84 EPHX2 (0.39) P2RX7EPHX2
SCHEMBL13191624 0.84 EPHX2 (0.40) P2RX7EPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010097373-A1 COMPOUNDS FOR USE AS BRADYKININ B1 ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-09-02 WO disclosed