Trifluoroacetic Acid

Trifluoroacetic Acid

SCHEMBL3725905

COc1ccc(Oc2ccc(CNC(=O)C3(N)CC3)nc2)c(C(F)(F)F)c1.O=C(O)C(F)(F)F

nearest known ligand 0.41

Full drug profile on Sugi Atlas →

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 1/20 0.41
EPHX2 P34913 8/20 0.39
ADORA2A P29274 1/20 0.38
PPARG P37231 3/20 0.37
KMT2A Q03164 2/20 0.36
MAPK8 P45983 1/20 0.35
MAPK10 P53779 1/20 0.35
ESRRA P11474 1/20 0.35
MEN1 O00255 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3719008 0.96 P2RX7 (0.43) P2RX7EPHX2ADORA2AKMT2AMAPK8
Trifluoroacetic Acid SCHEMBL2541472 0.88 HDAC3 (0.43) EPHX2PPARG
SCHEMBL3722862 0.87 P2RX7 (0.43) P2RX7EPHX2MAPK8MAPK10ESRRA
Trifluoroacetic Acid SCHEMBL2788039 0.84 L3MBTL1 (0.41) EPHX2PPARG
SCHEMBL2549180 0.84 L3MBTL1 (0.45) P2RX7EPHX2
SCHEMBL13191685 0.83 P2RX7 (0.39) P2RX7EPHX2ADORA2AKMT2AMAPK8
Trifluoroacetic Acid SCHEMBL2789689 0.83 P2RX7 (0.42) P2RX7EPHX2PPARG
SCHEMBL13191703 0.82 P2RX7 (0.38) P2RX7EPHX2ADORA2AKMT2AMEN1
SCHEMBL13191622 0.82 EPHX2 (0.47) P2RX7EPHX2PPARGKMT2AMEN1
SCHEMBL13191684 0.81 EPHX2 (0.39) P2RX7EPHX2PPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010097373-A1 COMPOUNDS FOR USE AS BRADYKININ B1 ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-09-02 WO disclosed