SCHEMBL3719115

SCHEMBL3719115

O=C(O)Cc1cnnc2ncncc12

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.33
MAPT P10636 2/20 0.33
CYP1A2 P05177 1/20 0.33
ALDH1A1 P00352 2/20 0.32
GABRA1 P14867 2/20 0.32
GABRA5 P31644 2/20 0.32
GABRB2 P47870 2/20 0.32
GABRA4 P48169 2/20 0.32
CYP3A4 P08684 1/20 0.32
TSHR P16473 1/20 0.32
NFKB1 P19838 1/20 0.32
GABRR1 P24046 1/20 0.32
GABRR2 P28476 1/20 0.32
PMP22 Q01453 1/20 0.31
NAPRT Q6XQN6 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
AKR1B1 P15121 1/20 0.31
PTGDR2 Q9Y5Y4 4/20 0.31
GABRP O00591 1/20 0.30
GABRD O14764 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3721023 0.80 DPP4 (0.43) KDM4EMAPTALDH1A1TSHRTDP1
SCHEMBL27350686 0.71 TDP1 (0.49) KDM4EMAPTCYP1A2ALDH1A1TDP1
SCHEMBL9431109 0.70 PIK3CG (0.33)
SCHEMBL479502 0.68 CYP2C19 (0.37) KDM4EMAPTALDH1A1GABRA1GABRA5
SCHEMBL12436875 0.67 GABRA5 (0.42) KDM4EMAPTCYP1A2ALDH1A1GABRA1
SCHEMBL907669 0.67 KDM4E (0.37) KDM4EMAPTCYP1A2ALDH1A1GABRA1
SCHEMBL3720458 0.67 MEN1 (0.38) KDM4EMAPTCYP1A2ALDH1A1
SCHEMBL3719119 0.65 GABRA5 (0.33) KDM4EMAPTALDH1A1GABRA1GABRA5
SCHEMBL27845043 0.63 AGBL2 (0.41) KDM4EMAPTCYP1A2ALDH1A1GABRA1
SCHEMBL907750 0.63 HSD17B10 (0.39) KDM4EMAPTCYP1A2ALDH1A1GABRA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010125469-A1 PYRIMIDINEDIONE-FUSED HETEROCYCLIC COMPOUNDS AS TRPA1 MODULATORS GLENMARK PHARMACEUTICALS, S.A. (CH) 2010-11-04 WO disclosed