SCHEMBL3720366

SCHEMBL3720366

NC(=O)c1cccc(-c2ccc(OCC(F)(F)F)cc2)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 1/20 0.50
FYN P06241 1/20 0.49
MAOB P27338 2/20 0.49
ABL1 P00519 3/20 0.47
RORC P51449 1/20 0.47
ERN1 O75460 2/20 0.47
PDK2 Q15119 1/20 0.47
PLG P00747 1/20 0.46
PLAU P00749 1/20 0.46
PLAT P00750 1/20 0.46
KDM4E B2RXH2 1/20 0.46
MAPT P10636 1/20 0.46
BCR P11274 1/20 0.46
MAPK1 P28482 1/20 0.46
SYK P43405 1/20 0.46
RXRA P19793 1/20 0.44
NR1H2 P55055 1/20 0.44
NR1H3 Q13133 1/20 0.44
FAAH O00519 1/20 0.44
DRD3 P35462 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15036779 0.84 PARP1 (0.56) MAOBKDM4EMAPT
SCHEMBL3721809 0.81 ABL1 (0.62) DHODHABL1ERN1PDK2PLAU
SCHEMBL6523003 0.80 MAOB (0.62) MAOBMAPT
SCHEMBL3717850 0.79 DHODH (0.74) DHODHERN1PDK2PLGPLAU
SCHEMBL28105217 0.79 KDR (0.58) DHODHABL1RORCERN1PDK2
SCHEMBL1787718 0.79 FYN (0.50) DHODHFYNERN1PLAUPLAT
SCHEMBL1787423 0.79 FYN (0.50) DHODHFYNERN1PLAUPLAT
Hydrochloric Acid SCHEMBL3722990 0.78 DHODH (0.72) DHODHERN1PDK2PLGPLAU
SCHEMBL6999225 0.76 DHODH (0.63) DHODHERN1MAPT
SCHEMBL3720494 0.76 PARP1 (0.67) ABL1PLGPLAUPLATKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8614201-B2 Heterocyclic amides as modulators of TRPA1 JANSSEN PHARMACEUTICA NV (BE) 2013-12-24 US claimed
WO-2010141805-A1 HETEROCYCLIC AMIDES AS MODULATORS OF TRPA1 JANSSEN PHARMACEUTICA NV (BE) 2010-12-09 WO claimed
US-8614201-B2 Heterocyclic amides as modulators of TRPA1 JANSSEN PHARMACEUTICA NV (BE) 2013-12-24 US disclosed
WO-2010141805-A1 HETEROCYCLIC AMIDES AS MODULATORS OF TRPA1 JANSSEN PHARMACEUTICA NV (BE) 2010-12-09 WO disclosed